PD 173212

PD 173212 is an N-type calcium channel blocker (IC50 = 36 nM). It prevents audiogenic seizures in mice when administered at a dose of 30 mg/kg.Formal Name: N-[[4-(1,1-dimethylethyl)phenyl]methyl]-N-methyl-L-leucyl-N-(1,1-dimethylethyl)-O-(phenylmethyl)-L-tyrosinamide. CAS Number: 217171-01-2. Molecular Formula: C38H53N3O3. Formula Weight: 599.9. Purity: >95%. Formulation: (Request formulation change), A solid. Solubility: DMSO: 100 mM, Ethanol: 100 mM. SMILES: CC(C)(C)C1=CC=C(CN(C)[C@@H](CC(C)C)C(N[C@@H](CC2=CC=C(OCC3=CC=CC=C3)C=C2)C(NC(C)(C)C)=O)=O)C=C1. InChi Code: InChI=1S/C38H53N3O3/c1-27(2)23-34(41(9)25-29-15-19-31(20-16-29)37(3,4)5)36(43)39-33(35(42)40-38(6,7)8)24-28-17-21-32(22-18-28)44-26-30-13-11-10-12-14-30/h10-22,27,33-34H,23-26H2,1-9H3,(H,39,43)(H,40,42)/t33-,34-/m0/s1. InChi Key: GCDHMGROXQUFNR-HEVIKAOCSA-N.