Masofaniten

Masofaniten is an androgen receptor N-terminal transactivation domain inhibitor (ARTADI). It binds to the tryptophan residues in positions 397 (W397) and W433 in the AR TAD.Formal Name: N-[4-[[4-[1-[3-chloro-4-(2-chloroethoxy)-5-cyanophenyl]-1-methylethyl]phenoxy]methyl]-2-pyrimidinyl]-methanesulfonamide. CAS Number: 2416716-62-4. Synonyms: EPI-7386. Molecular Formula: C24H24Cl2N4O4S. Formula Weight: 535.4. Purity: >95%. Formulation: (Request formulation change), A solid. Solubility: DMSO: Sparingly soluble: 1-10 mg/ml. SMILES: N#CC1=CC(C(C)(C)C2=CC=C(C=C2)OCC3=NC(NS(=O)(C)=O)=NC=C3)=CC(Cl)=C1OCCCl. InChi Code: InChI=1S/C24H24Cl2N4O4S/c1-24(2,18-12-16(14-27)22(21(26)13-18)33-11-9-25)17-4-6-20(7-5-17)34-15-19-8-10-28-23(29-19)30-35(3,31)32/h4-8,10,12-13H,9,11,15H2,1-3H3,(H,28,29,30). InChi Key: GVCZSODXLFBYSS-UHFFFAOYSA-N.