I-BET762

Item number	Size	Manual	SDS	Delivery time	Price
SYN-3033-M001	1 mg	-	-	3 - 9 business days*	123.00€
SYN-3033-M005	5 mg	-	-	3 - 9 business days*	185.00€
SYN-3033-M010	10 mg	-	-	3 - 9 business days*	246.00€
SYN-3033-M050	50 mg	-	-	3 - 9 business days*	693.00€
SYN-3033-M100	100 mg	-	-	3 - 9 business days*	1,109.00€

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I-BET762 (GSK525762A) is an inhibitor for BET (bromodomain and extra terminal domain) proteins,... more

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Product information "I-BET762"

I-BET762 (GSK525762A) is an inhibitor for BET (bromodomain and extra terminal domain) proteins, BRD2, BRD3 and BRD4. It binds to the tandem bromodomains of BET with a Kd of 50.5-61.3nM, displaces a tetra-acetylated H4 peptide prebound to tandem bromodomains of BET with IC50 of 32.5-42.5nM in FRET analysis. I-BET762 disrupts the formation of the chromatin complexes essential for expression of inflammatory genes.

Keywords:	GSK-525762A
Supplier:	SYNkinase
Supplier-Nr:	3033

Properties

Application:	BET (bromodomain and extra terminal domain) protein BRD2 / BRD3 / BRD4 inhibitor
MW:	423.9 D
Formula:	C22H22ClN5O2
Purity:	>95%
Format:	Solid

Database Information

CAS :	1260907-17-2\| Matching products
KEGG ID :	K08871 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+20°C (International: +20°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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