I-BET151 (GSK1210151A)

Item number	Size	Manual	SDS	Delivery time	Price
BPS-27629-1	5 mg	-	-	3 - 15 business days*	410.00€
BPS-27629-2	10 mg	-	-	3 - 15 business days*	464.00€
BPS-27629-3	50 mg	-	-	3 - 15 business days*	943.00€

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I-BET151(GSK1210151A) is a BET bromodomain inhibitor. I-BET151 displays potent binding affinity... more

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Product information "I-BET151 (GSK1210151A)"

I-BET151(GSK1210151A) is a BET bromodomain inhibitor. I-BET151 displays potent binding affinity to BRD2, BRD3 and BRD4 with Kd of 0.02-0.1 µM. I-BET151 (0.5 or 5 µM) inhibits the binding of BETs (BRD2, BRD3, BRD4, and BRD9) but not the binding of 23 other bromodomain proteins. I-BET151 also blocks recruitment of BET to chromatin.

Keywords:	I-BET151, GSK1210151A, 7-(3,5-dimethyl-1,2-oxazol-4-yl)-8-methoxy-1-[(1R)-1-pyridin-2-ylethyl]-3H-imidazo[4,5-c]quinolin-2-one,
Supplier:	BPS Bioscience
Supplier-Nr:	27629