GSK343
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: GSK343, a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold... more
Product information "GSK343"
Description: GSK343, a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold specificity activity against EZH1, and >1000 fold specificity activity against other histone methyltransferases. Target: Histone Methyltransferase, Autophagy. Smiles: CCCc1cc(C)[nH]c(=O)c1CNC(=O)c1cc(cc2n(ncc12)C(C)C)-c1ccnc(c1)N1CCN(C)CC1. References: Verma SK, et al. ACS Med Chem Lett. 2012, 3, 1091-1096.
| Supplier: | TargetMol |
| Supplier-Nr: | T6059 |
Properties
| Application: | Cell-permeable EZH2 inhibitor |
| MW: | 541.69 D |
| Formula: | C31H39N7O2 |
Database Information
| CAS : | 1346704-33-3| Matching products |
| KEGG ID : | K11430 | Matching products |
Handling & Safety
| Storage: | +4°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H302 |
| P Phrases: | P264, P270, P301+310, P330, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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