GSK180736A

Item number	Size	Delivery time	Price
TGM-T3513-1mg	1 mg	7 - 10 business days*	37.00€
TGM-T3513-2mg	2 mg	7 - 10 business days*	48.00€
TGM-T3513-1mL	1 ml	7 - 10 business days*	60.00€
TGM-T3513-5mg	5 mg	7 - 10 business days*	67.00€
TGM-T3513-10mg	10 mg	7 - 10 business days*	89.00€
TGM-T3513-25mg	25 mg	7 - 10 business days*	172.00€
TGM-T3513-50mg	50 mg	7 - 10 business days*	322.00€
TGM-T3513-100mg	100 mg	7 - 10 business days*	597.00€
TGM-T3513-500mg	500 mg	7 - 10 business days*	1,289.00€

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Description: GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 µM) and... more

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Product information "GSK180736A"

Description: GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 µM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 µM), but highly effective against ROCK1 (IC50: 100 nM). Target: ROCK, GRK, PKA. Smiles: CC1=C(C(NC(=O)N1)c1ccc(F)cc1)C(=O)Nc1ccc2[nH]ncc2c1. References: Homan KT, et al. ACS Chem Biol. 2015, 10(1):310-9.

Keywords:	GSK180736
Supplier:	TargetMol
Supplier-Nr:	T3513

Properties

Application:	ROCK1 inhibitor
MW:	365.36 D
Formula:	C19H16FN5O2

Database Information

CAS :	817194-38-0\| Matching products
KEGG ID :	K04514 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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