GSK126

Item number	Size	Delivery time	Price
TGM-T2079-2mg	2 mg	7 - 10 business days*	39.00€
TGM-T2079-5mg	5 mg	7 - 10 business days*	59.00€
TGM-T2079-1mL	1 ml	7 - 10 business days*	68.00€
TGM-T2079-10mg	10 mg	7 - 10 business days*	90.00€
TGM-T2079-25mg	25 mg	7 - 10 business days*	156.00€
TGM-T2079-50mg	50 mg	7 - 10 business days*	239.00€
TGM-T2079-100mg	100 mg	7 - 10 business days*	374.00€
TGM-T2079-200mg	200 mg	7 - 10 business days*	488.00€

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Description: GSK126 (GSK2816126A) is a excellently specific EZH2 methyltransferase inhibitor (... more

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Product information "GSK126"

Description: GSK126 (GSK2816126A) is a excellently specific EZH2 methyltransferase inhibitor ( IC50=9.9 nM). Target: Histone Methyltransferase. Smiles: CC[C@H](C)n1cc(C)c2c(cc(cc12)-c1ccc(nc1)N1CCNCC1)C(=O)NCc1c(C)cc(C)[nH]c1=O. References: Ott HM, et al. A687V EZH2 is a driver of histone H3 lysine 27 (H3K27) hypertrimethylation. Mol Cancer Ther. 2014 Dec,13(12):3062-73.

Keywords:	GSK2816126A, EZH2 inhibitor
Supplier:	TargetMol
Supplier-Nr:	T2079

Properties

Application:	Selective EZH2 methyltransferase inhibitor
MW:	526.67 D
Formula:	C31H38N6O2

Database Information

CAS :	1346574-57-9\| Matching products
KEGG ID :	K11430 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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