GSK-5959

Item number	Size	Delivery time	Price
TGM-T1972-5mg	5 mg	7 - 10 business days*	52.00€
TGM-T1972-1mL	1 ml	7 - 10 business days*	58.00€
TGM-T1972-10mg	10 mg	7 - 10 business days*	88.00€
TGM-T1972-25mg	25 mg	7 - 10 business days*	159.00€
TGM-T1972-50mg	50 mg	7 - 10 business days*	261.00€
TGM-T1972-100mg	100 mg	7 - 10 business days*	390.00€
TGM-T1972-200mg	200 mg	7 - 10 business days*	571.00€

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Description: GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor... more

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Product information "GSK-5959"

Description: GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Target: Epigenetic Reader Domain. Smiles: COc1ccccc1C(=O)Nc1cc2n(C)c(=O)n(C)c2cc1N1CCCCC1. References: Demont EH, et al. ACS Med Chem Lett. 5(11):1190-1195.

Supplier:	TargetMol
Supplier-Nr:	T1972

Properties

Application:	BRPF1 (Peregrin) bromodomain inhibitor
MW:	394.47 D
Formula:	C22H26N4O3

Database Information

CAS :	901245-65-6\| Matching products
KEGG ID :	K11348 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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