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GNE-781

TargetMol
GNE-781
Item number Size Datasheet Manual SDS Delivery time Quantity Price
TGM-T15405-1mg 1 mg

7 - 10 business days*

168.00€
TGM-T15405-5mg 5 mg

7 - 10 business days*

371.00€
TGM-T15405-1mL 1 ml

7 - 10 business days*

419.00€
TGM-T15405-10mg 10 mg

7 - 10 business days*

566.00€
TGM-T15405-25mg 25 mg

7 - 10 business days*

914.00€
TGM-T15405-50mg 50 mg

7 - 10 business days*

1,244.00€
TGM-T15405-100mg 100 mg

7 - 10 business days*

1,684.00€
If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
 
Description Product Citations Certificate of Analysis Reviews 0
Description
Description: GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET... more
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Product information "GNE-781"
Description: GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay). GNE-781 also inhibits BRET and BRD4(1) (IC50s: 6.2 nM and 5100 nM, respectively). Target: Epigenetic Reader Domain. Smiles: CNC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)N1CCCc2cc(-c3cnn(C)c3)c(cc12)C(F)F. References: Romero FA, et al. GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP). J Med Chem. 2017 Nov 22,60(22):9162-9183.
Supplier: TargetMol
Supplier-Nr: T15405

Properties

Application: CBP / p300 inhibitor
MW: 525.59 D
Formula: C27H33F2N7O2

Database Information

CAS : 1936422-33-1| Matching products
KEGG ID : K04498 | Matching products

Handling & Safety

Storage: +4°C
Shipping: +4°C (International: +4°C)
Caution
Our products are for laboratory research use only: Not for administration to humans!
Product Citations
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