Gilteritinib

Item number	Size	Delivery time	Price
TGM-T4409-1mg	1 mg	7 - 10 business days*	34.00€
TGM-T4409-2mg	2 mg	7 - 10 business days*	50.00€
TGM-T4409-5mg	5 mg	7 - 10 business days*	80.00€
TGM-T4409-10mg	10 mg	7 - 10 business days*	120.00€
TGM-T4409-25mg	25 mg	7 - 10 business days*	192.00€
TGM-T4409-50mg	50 mg	7 - 10 business days*	284.00€
TGM-T4409-100mg	100 mg	7 - 10 business days*	447.00€
TGM-T4409-500mg	500 mg	7 - 10 business days*	1,039.00€
TGM-T4409-1g	1 g	7 - 10 business days*	1,402.00€

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Description: Gilteritinib (ASP2215) is a potent inhibitor of FMS-related tyrosine kinase 3 (FLT3)... more

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Product information "Gilteritinib"

Description: Gilteritinib (ASP2215) is a potent inhibitor of FMS-related tyrosine kinase 3 (FLT3) and AXL tyrosine kinase receptors (IC50 = 0.29 nM and <1 nM, respectively). In preclinical studies, gilteritinib demonstrated strong antileukemic and antitumor effects. Gilteritinib is currently in several Phase 3 clinical trials for acute myeloid leukemia. Target: TAM Receptor, c-Kit, FLT. Smiles: CCc1nc(C(N)=O)c(Nc2ccc(N3CCC(CC3)N3CCN(C)CC3)c(OC)c2)nc1NC1CCOCC1. References: Mori M, et al. Gilteritinib, a FLT3/AXL inhibitor, shows antileukemic activity in mouse models of FLT3 mutated acute myeloid leukemia. Invest New Drugs. 2017 Oct,35(5):556-565.

Keywords:	ASP2215
Supplier:	TargetMol
Supplier-Nr:	T4409

Properties

Application:	Targets fms-related tyrosine kinase 3 [EC:2.7.10.1] (FLT3, FLK2, CD135)
MW:	552.71 D
Formula:	C29H44N8O3

Database Information

CAS :	1254053-43-4\| Matching products
KEGG ID :	K05092 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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