Gemfibrozil 1-O-beta-glucuronide

Item number	Size	Datasheet	Manual	SDS	Delivery time	Quantity	Price
TGM-T11387-500ug	500 µg		-		7 - 10 business days*		592.00€
TGM-T11387-1mg	1 mg				7 - 10 business days*		1,140.00€

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Description: Gemfibrozil 1-O-beta-Glucuronide, a metabolite of Gemfibrozil, is a potent and... more

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Product information "Gemfibrozil 1-O-beta-glucuronide"

Description: Gemfibrozil 1-O-beta-Glucuronide, a metabolite of Gemfibrozil, is a potent and competitive inhibitor of P450 (CYP) isoform CYP2C8, with an IC50 of 4.07 µM. Target: Others. Smiles: Cc1ccc(C)c(OCCCC(C)(C)C(=O)O[C@@H]2O[C@@H]([C@@H](O)[C@H](O)[C@H]2O)C(O)=O)c1. References: Shitara Y, et al. Gemfibrozil and its glucuronide inhibit the organic anion transporting polypeptide 2(OATP2/OATP1B1:SLC21A6)-mediated hepatic uptake and CYP2C8-mediated metabolism of cerivastatin: analysis of the mechanism of the clinically relevant drug-drug interaction between cerivastatin and gemfibrozil. J Pharmacol Exp Ther. 2004 Oct,311(1):228-36.

Supplier:	TargetMol
Supplier-Nr:	T11387

Properties

MW:	426.46 D
Formula:	C21H30O9

Database Information

CAS :

91683-38-4| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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