ERK1/2 inhibitor 1

Item number	Size	Delivery time	Price
TGM-T11226-1mg	1 mg	7 - 10 business days*	128.00€
TGM-T11226-5mg	5 mg	7 - 10 business days*	320.00€
TGM-T11226-1mL	1 ml	7 - 10 business days*	355.00€
TGM-T11226-10mg	10 mg	7 - 10 business days*	464.00€
TGM-T11226-25mg	25 mg	7 - 10 business days*	712.00€
TGM-T11226-50mg	50 mg	7 - 10 business days*	952.00€
TGM-T11226-100mg	100 mg	7 - 10 business days*	1,300.00€

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Description: ERK1/2 inhibitor 1 is a potent, orally bioavailable compound that exhibits 60%... more

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Product information "ERK1/2 inhibitor 1"

Description: ERK1/2 inhibitor 1 is a potent, orally bioavailable compound that exhibits 60% inhibition at 1 nM and has an IC50 of 3.0 nM against ERK1 and ERK2, respectively. Target: ERK. Smiles: C[C@@H](N1Cc2ccc(cc2C1=O)-c1nc(NC2CCOCC2)ncc1Cl)C(=O)N[C@H](CO)c1cccc(C)c1. References: Heightman TD, et al. Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2. J Med Chem. 2018 Jun 14,61(11):4978-4992.

Supplier:	TargetMol
Supplier-Nr:	T11226

Properties

Application:	ERK1/2 inhibitor
MW:	550.05 D
Formula:	C29H32ClN5O4

Database Information

CAS :	2095719-90-5\| Matching products
KEGG ID :	K04371 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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