Enzalutamide
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP)... more
Product information "Enzalutamide"
Description: Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP) that activates autophagy, exhibits antitumor activity, and is commonly used in treating desmoplasia-resistant prostate cancer. Target: Autophagy, Androgen Receptor. Smiles: S=C1N(C(C)(C)C(=O)N1C2=CC(C(F)(F)F)=C(C#N)C=C2)C3=CC(F)=C(C(NC)=O)C=C3. References: Wright TC, et al. Abiraterone In Vitro Is Superior to Enzalutamide in Response to Ionizing Radiation. Front Oncol. 2021 Jul 21,11:700543.
| Keywords: | MDV3100 |
| Supplier: | TargetMol |
| Supplier-Nr: | T6002 |
Properties
| Application: | Targets androgen receptor (AR, NR3C4) |
| MW: | 464.44 D |
| Formula: | C21H16F4N4O2S |
Database Information
| CAS : | 915087-33-1| Matching products |
| KEGG ID : | K08557 | Matching products |
| Protein Atlas Nr. : | Gene Regulation |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H361 |
| P Phrases: | P201, P202, P280, P308+313, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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