Entrectinib

Item number	Size	Delivery time	Price
TGM-T3678-2mg	2 mg	7 - 10 business days*	37.00€
TGM-T3678-5mg	5 mg	7 - 10 business days*	55.00€
TGM-T3678-1mL	1 ml	7 - 10 business days*	62.00€
TGM-T3678-10mg	10 mg	7 - 10 business days*	81.00€
TGM-T3678-25mg	25 mg	7 - 10 business days*	112.00€
TGM-T3678-50mg	50 mg	7 - 10 business days*	170.00€
TGM-T3678-100mg	100 mg	7 - 10 business days*	295.00€
TGM-T3678-500mg	500 mg	7 - 10 business days*	727.00€

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Description: Entrectinib (RXDX-101) is a Trk, ROS1, and ALK inhibitor that inhibits TrkA, TrkB,... more

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Product information "Entrectinib"

Description: Entrectinib (RXDX-101) is a Trk, ROS1, and ALK inhibitor that inhibits TrkA, TrkB, TrkC, ROS1, and ALK (IC50=1/3/5/12/7 nM) with oral activity and blood-brain-barrier penetration. Entrectinib exhibits both antitumor and CNS activity. Target: ALK, ROS Kinase, ROS, Autophagy, Trk receptor. Smiles: N(C(=O)C1=C(NC2CCOCC2)C=C(C=C1)N3CCN(C)CC3)C=4C=5C(NN4)=CC=C(CC6=CC(F)=CC(F)=C6)C5. References: Rolfo C, et al. Expert Opin Investig Drugs. 2015, 24(11), 1493-1500.

Keywords:	RXDX-101, NMS-E628
Supplier:	TargetMol
Supplier-Nr:	T3678

Properties

Application:	Targets neurotrophic tyrosine kinase receptor type 1 [EC:2.7.10.1] (NTRK1, TRKA)
MW:	560.64 D
Formula:	C31H34F2N6O2

Database Information

CAS :	1108743-60-7\| Matching products
KEGG ID :	K03176 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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