Ensifentrine

Item number	Size	Delivery time	Price
TGM-T25376-1mg	1 mg	7 - 10 business days*	31.00€
TGM-T25376-5mg	5 mg	7 - 10 business days*	97.00€
TGM-T25376-1mL	1 ml	7 - 10 business days*	106.00€
TGM-T25376-10mg	10 mg	7 - 10 business days*	161.00€
TGM-T25376-25mg	25 mg	7 - 10 business days*	345.00€
TGM-T25376-50mg	50 mg	7 - 10 business days*	560.00€
TGM-T25376-100mg	100 mg	7 - 10 business days*	891.00€

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Description: Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for... more

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Product information "Ensifentrine"

Description: Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3(IC50: 0.4 nM) is 3,440 times higher than that for PDE4(IC50: 1479 nM), that is under clinical development for the treatment of asthma and COPD and, potentially, cystic fibrosis. Target: PDE. Smiles: COc1cc2CCn3c(c\c(=N/c4c(C)cc(C)cc4C)n(CCNC(N)=O)c3=O)-c2cc1OC. References: Henrik Watz, et al. Symptom Improvement Following Treatment with the Inhaled Dual Phosphodiesterase 3 and 4 Inhibitor Ensifentrine in Patients with Moderate to Severe COPD - A Detailed Analysis. Int J Chron Obstruct Pulmon Dis. 2020 Sep 16,15:2199-2206.

Keywords:	Ensifentrinum, Ensifentrina
Supplier:	TargetMol
Supplier-Nr:	T25376

Properties

Application:	Targets cAMP-specific phosphodiesterase 4 [EC:3.1.4.53] (PDE4)
MW:	477.56 D
Formula:	C26H31N5O4
Format:	32160405

Database Information

CAS :	1884461-72-6\| Matching products
KEGG ID :	K13293 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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