Dimaprit (hydrochloride)

Dimaprit (hydrochloride)
Item number Size Datasheet Manual SDS Delivery time Quantity Price
Cay29418-50 50 mg -

6 - 10 business days*

90.00€
Cay29418-100 100 mg -

6 - 10 business days*

143.00€
Cay29418-250 250 mg -

6 - 10 business days*

333.00€
 
Dimaprit is a histamine H2 receptor agonist with a Ki value of 44 µM in guinea pig right atrium.... more
Product information "Dimaprit (hydrochloride)"
Dimaprit is a histamine H2 receptor agonist with a Ki value of 44 µM in guinea pig right atrium. It is selective for histamine H2 over H1 and H3 receptors with relative potencies of 71, A. suum extract, which is not affected by pretreatment with mepyramine (Cay-20978), an H1 receptor inverse agonist, or cimetidine (Cay-18743), an H2 receptor antagonist. It stimulates gastric acid secretion in vivo in anaesthetized rats and cats with relative potencies of 19.5 and approximately 400 to 500, respectively, compared to histamine. Dimaprit inhibits 2-(2-pyridyl)ethylamine-induced bronchoconstriction in guinea pigs in a dose-dependent manner.Formal Name: carbamimidothioic acid, 3-(dimethylamino)propyl ester, dihydrochloride. CAS Number: 23256-33-9. Molecular Formula: C6H15N3S . 2HCl. Formula Weight: 234.2. Purity: >95%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 30 mg/ml, DMSO: 30 mg/ml, DMSO:PBS (pH 7.2) (1:3): 0.25 mg/ml. SMILES: NC(SCCCN(C)C)=N.Cl.Cl. InChi Code: InChI=1S/C6H15N3S.2ClH/c1-9(2)4-3-5-10-6(7)8,,/h3-5H2,1-2H3,(H3,7,8),2*1H. InChi Key: DFWCPLGXFMSUCW-UHFFFAOYSA-N.
Keywords: carbamimidothioic acid, 3-(dimethylamino)propyl ester, dihydrochloride
Supplier: Cayman Chemical
Supplier-Nr: 29418

Properties

Application: Histamine H2 receptor agonist
MW: 234.2 D
Formula: C6H15N3S . 2HCl
Purity: >95%
Format: Crystalline Solid

Database Information

CAS : 23256-33-9| Matching products
KEGG ID : K04150 | Matching products

Handling & Safety

Storage: -20°C
Shipping: +20°C (International: -20°C)
Signal Word: Warning
GHS Hazard Pictograms:
H Phrases: H315, H319, H335
P Phrases: P261, P264, P271, P280, P302+352, P304+340, P305+351+338, P312, P321, P332+313, P337+313, P362+364, P403+233, P405, P501
Caution
Our products are for laboratory research use only: Not for administration to humans!
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