Darapladib
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You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: Darapladib (SB-480848)(IC50=0.25 nM) is a substituted pyrimidone with inhibitory... more
Product information "Darapladib"
Description: Darapladib (SB-480848)(IC50=0.25 nM) is a substituted pyrimidone with inhibitory activity towards lipoprotein-associated phospholipase-A2 (Lp-PLA2). Target: Phospholipase. Smiles: C(C(N(CC1=CC=C(C=C1)C2=CC=C(C(F)(F)F)C=C2)CCN(CC)CC)=O)N3C4=C(C(=O)N=C3SCC5=CC=C(F)C=C5)CCC4. References: Blackie JA, et al. Bioorg Med Chem Lett. 2003, 13(6), 1067-1070.
| Keywords: | SB-480848 |
| Supplier: | TargetMol |
| Supplier-Nr: | T6109 |
Properties
| Application: | Targets platelet-activating factor acetylhydrolase [EC:3.1.1.47] (PLA2G7, PAFAH) |
| MW: | 666.77 D |
| Formula: | C36H38F4N4O2S |
Database Information
| CAS : | 356057-34-6| Matching products |
| KEGG ID : | K01062 | Matching products |
| Protein Atlas Nr. : | Metabolism |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Danger |
| GHS Hazard Pictograms: |
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| H Phrases: | H318, H400, H410 |
| P Phrases: | P273, P280, P310, P391, P305+P351+P338, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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