CYC-116

Item number	Size	Delivery time	Price
TGM-T6458-2mg	2 mg	7 - 10 business days*	33.00€
TGM-T6458-1mL	1 ml	7 - 10 business days*	45.00€
TGM-T6458-5mg	5 mg	7 - 10 business days*	51.00€
TGM-T6458-10mg	10 mg	7 - 10 business days*	70.00€
TGM-T6458-25mg	25 mg	7 - 10 business days*	134.00€
TGM-T6458-50mg	50 mg	7 - 10 business days*	224.00€
TGM-T6458-100mg	100 mg	7 - 10 business days*	368.00€
TGM-T6458-500mg	500 mg	7 - 10 business days*	936.00€

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Description: CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent... more

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Product information "CYC-116"

Description: CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent to VEGFR2 (Ki of 44 nM), with 50-fold greater potency than CDKs, not active against PKA, Akt/PKB, PKC, no effect on GSK-3alpha/beta, CK2, Plk1 and SAPK2A. Phase 1. Target: FLT, CDK, Aurora Kinase, VEGFR, S6 Kinase. Smiles: Cc1nc(N)sc1-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1. References: Wang S, et al. J Med Chem. 2010, 53(11), 4367-4378.

Supplier:	TargetMol
Supplier-Nr:	T6458

Properties

MW:	368.46 D
Formula:	C18H20N6OS

Database Information

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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