CVT-2738

CVT-2738 is an active metabolite of the antianginal agent ranolazine (Cay-15604). It is formed from ranolazine by the cytochrome P450 (CYP) isoform CYP3A. CVT-2738 (100 mg/kg) inhibits increases in T-wave height and the RR interval in a mouse model of myocardial ischemia induced by isoprenaline (isoproterenol, Cay-15592).Formal Name: N-(2,6-dimethylphenyl)-1-piperazineacetamide. CAS Number: 5294-61-1. Molecular Formula: C14H21N3O. Formula Weight: 247.3. Purity: >98%. Formulation: (Request formulation change), A solid. Solubility: DMF: 10 mg/ml, DMF:PBS (pH 7.2) (1:5): 0.16 mg/ml, DMSO: 5 mg/ml, Ethanol: 5 mg/ml. SMILES: O=C(CN1CCNCC1)NC2=C(C)C=CC=C2C. InChi Code: InChI=1S/C14H21N3O/c1-11-4-3-5-12(2)14(11)16-13(18)10-17-8-6-15-7-9-17/h3-5,15H,6-10H2,1-2H3,(H,16,18). InChi Key: NJKRFQIWDJSYOK-UHFFFAOYSA-N.