CAY10789

Item number	Size	Delivery time	Price
TGM-T60439-1mg	1 mg	7 - 10 business days*	110.00€
TGM-T60439-5mg	5 mg	7 - 10 business days*	476.00€
TGM-T60439-10mg	10 mg	7 - 10 business days*	784.00€
TGM-T60439-25mg	25 mg	7 - 10 business days*	1,674.00€

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Description: CAY10789 (compound 6) is a potent CysLT1R (cysteinyl leukotriene receptor 1)... more

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Product information "CAY10789"

Description: CAY10789 (compound 6) is a potent CysLT1R (cysteinyl leukotriene receptor 1) antagonist with an IC50 of 2.80 µM and a GPBAR1 (G-protein-coupled bile acid receptor 1) agonist with an EC50 of 3 µM. It significantly decreases U937 cell adhesion to HAEC and reduces TNF-alpha expression. CAY10789 demonstrates promising metabolic stability and excellent pharmacokinetics, making it suitable for studying colitis, metabolic syndromes, and other GPBAR1/CysLT1R-related diseases [1]. Target: Others. Smiles: C(OC1=CC(CO)=CC=C1)C2=NC3=C(C=C2)C=CC=C3

Supplier:	TargetMol
Supplier-Nr:	T60439

Properties

Application:	CysLT1 receptor antagonist
MW:	265.31 D
Formula:	C17H15NO2

Database Information

CAS :	123226-28-8\| Matching products
KEGG ID :	K04322 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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