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![Bupivacaine](https://www.biomol.com/media/image/64/70/b6/Cay16618-1_600x600.png)
Item number | Size | Datasheet | Manual | SDS | Delivery time | Quantity | Price |
---|---|---|---|---|---|---|---|
Cay16618-500 | 500 mg | - |
6 - 10 business days* |
43.00€
|
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Cay16618-1 | 1 g | - |
6 - 10 business days* |
68.00€
|
If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Bupivacaine is a sodium channel blocker and local anesthetic. It inhibits sodium currents in rat... more
Product information "Bupivacaine"
Bupivacaine is a sodium channel blocker and local anesthetic. It inhibits sodium currents in rat dorsal horn neurons in a concentration-dependent manner and inhibits synaptic transmission in rat sympathetic ganglia, increasing the firing threshold when used at a concentration of 200 nM. Bupivacaine (10 µM) blocks cardiac sodium channels in a use-dependent manner and inhibits respiration in cardiac cell mitochondria when palmitoyl-carnitine or acetyl-carnitine are used as substrates (IC50s = 0.78 and 0.37 mM, respectively). It also reduces thermal hyperplasia in a rat model of sciatic ligation injury when 0.6 ml of a 0.5% solution is administered into the perinerve space, and the duration of this effect is extended by co-administration of the NMDA receptor antagonist MK-801 (Cay-10009019). Formulations containing bupivacaine have been used as local anesthetics for surgery, oral surgery, and dental procedures and for anesthetic purposes in research studies using animals.Formal Name: 1-butyl-N-(2,6-dimethylphenyl)-2-piperidinecarboxamide. CAS Number: 38396-39-3. Molecular Formula: C18H28N2O. Formula Weight: 288.4. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 30 mg/ml, DMSO: 25 mg/ml, Ethanol: 30 mg/ml, Ethanol:PBS(pH 7.2) (1:1): 0.5 mg/ml. SMILES: CC1=CC=CC(C)=C1NC(C2N(CCCC)CCCC2)=O. InChi Code: InChI=1S/C18H28N2O/c1-4-5-12-20-13-7-6-11-16(20)18(21)19-17-14(2)9-8-10-15(17)3/h8-10,16H,4-7,11-13H2,1-3H3,(H,19,21). InChi Key: LEBVLXFERQHONN-UHFFFAOYSA-N.
Keywords: | 1-butyl-N-(2,6-dimethylphenyl)-2-piperidinecarboxamide |
Supplier: | Cayman Chemical |
Supplier-Nr: | 16618 |
Properties
Application: | Sodium influx blocker |
MW: | 288.4 D |
Formula: | C18H28N2O |
Purity: | >98% |
Format: | Crystalline Solid |
Database Information
CAS : | 38396-39-3| Matching products |
KEGG ID : | K04841 | Matching products |
Handling & Safety
Storage: | -20°C |
Shipping: | +20°C (International: -20°C) |
Signal Word: | Danger |
GHS Hazard Pictograms: |
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H Phrases: | H300, H310, H330 |
P Phrases: | P260, P262, P264, P270, P271, P280, P284, P301+310, P302+352, P304+340, P310, P320, P321, P330, P361+364, P403+233, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
Information about the product reference will follow.
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