BRM/BRG1 ATP Inhibitor-1

Item number	Size	Manual	Delivery time	Price
TGM-T10616-1mg	1 mg	-	7 - 10 business days*	408.00€
TGM-T10616-1mL	1 ml	-	7 - 10 business days*	556.00€
TGM-T10616-5mg	5 mg	-	7 - 10 business days*	797.00€
TGM-T10616-10mg	10 mg	-	7 - 10 business days*	1,206.00€
TGM-T10616-25mg	25 mg	-	7 - 10 business days*	1,795.00€
TGM-T10616-50mg	50 mg	-	7 - 10 business days*	2,424.00€
TGM-T10616-100mg	100 mg	-	7 - 10 business days*	3,269.00€

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Description: BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related... more

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Product information "BRM/BRG1 ATP Inhibitor-1"

Description: BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A member 2 (SMARCA2) and BRG1/SMARCA4 ATPase activity inhibitor (IC50s<0.005 µM). Target: Epigenetic Reader Domain. Smiles: OCc1cnc(F)cc1NC(=O)Nc1cc(ns1)C(F)F. References: Papillon JPN, et al. Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers. J Med Chem. 2018 Nov 21,61(22):10155-10172

Supplier:	TargetMol
Supplier-Nr:	T10616

Properties

Application:	SMARCA2A/SMARCA4 ATPase inhibitor
MW:	318.27 D
Formula:	C11H9F3N4O2S

Database Information

CAS :	2270879-17-7\| Matching products
KEGG ID :	K11647 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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