Brepocitinib P-Tosylate

Item number	Size	Delivery time	Price
TGM-T12427-1mg	1 mg	7 - 10 business days*	31.00€
TGM-T12427-5mg	5 mg	7 - 10 business days*	63.00€
TGM-T12427-1mL	1 ml	7 - 10 business days*	79.00€
TGM-T12427-10mg	10 mg	7 - 10 business days*	105.00€
TGM-T12427-25mg	25 mg	7 - 10 business days*	228.00€
TGM-T12427-50mg	50 mg	7 - 10 business days*	411.00€
TGM-T12427-100mg	100 mg	7 - 10 business days*	660.00€

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Description: Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus... more

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Product information "Brepocitinib P-Tosylate"

Description: Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s of 17 nM and 23 nM, respectively). Target: JAK. Smiles: Cc1ccc(cc1)S(O)(=O)=O.Cn1cc(Nc2nccc(n2)N2CC3CCC(C2)N3C(=O)[C@@H]2CC2(F)F)cn1. References: Fensome A, et al. Dual Inhibition of TYK2 and JAK1 for the Treatment of Autoimmune Diseases: Discovery of (( S)-2,2-Difluorocyclopropyl)((1 R,5 S)-3-(2-((1-methyl-1 H-pyrazol-4-yl)amino)pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methanone (PF-06700841). J Med Chem. 2018 Oct 11,61(19):8597-8612.

Keywords:	PF-06700841 P-Tosylate
Supplier:	TargetMol
Supplier-Nr:	T12427

Properties

Application:	Targets Janus kinase 1 [EC:2.7.10.2] (JAK1)
MW:	561.6 D
Formula:	C25H29F2N7O4S
Format:	32160405

Database Information

CAS :	2140301-96-6\| Matching products
KEGG ID :	K11217 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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