Borussertib

Item number	Size	Manual	Delivery time	Price
TGM-T8427-1mg	1 mg	-	7 - 10 business days*	132.00€
TGM-T8427-5mg	5 mg	-	7 - 10 business days*	282.00€
TGM-T8427-1mL	1 ml	-	7 - 10 business days*	371.00€
TGM-T8427-10mg	10 mg	-	7 - 10 business days*	445.00€
TGM-T8427-25mg	25 mg	-	7 - 10 business days*	738.00€
TGM-T8427-50mg	50 mg	-	7 - 10 business days*	1,039.00€
TGM-T8427-100mg	100 mg	-	7 - 10 business days*	1,402.00€

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Description: Borussertib is a first-in-class covalent-allosteric inhibitor of protein kinase Akt,... more

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Product information "Borussertib"

Description: Borussertib is a first-in-class covalent-allosteric inhibitor of protein kinase Akt, with an IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt. Target: Akt. Smiles: C=CC(=O)Nc1ccc2[nH]c(=O)n(C3CCN(Cc4ccc(cc4)-c4nc5cc[nH]c(=O)c5cc4-c4ccccc4)CC3)c2c1. References: Niklas Uhlenbrock, et al. Structural and chemical insights into the covalentallosteric inhibition of the protein kinase Akt. Chem Sci., 2019, 10, 3573.

Supplier:	TargetMol
Supplier-Nr:	T8427

Properties

Application:	Akt1 / Akt2 inhibitor
MW:	596.68 D
Formula:	C36H32N6O3

Database Information

CAS :	1800070-77-2\| Matching products
KEGG ID :	K04456 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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