BMS-986122
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Larger quantity required? Request bulk
Description: BMS-986122 (BMS 986122) is a positive allosteric modulator of µ-opioid receptors... more
Product information "BMS-986122"
Description: BMS-986122 (BMS 986122) is a positive allosteric modulator of µ-opioid receptors that increases beta-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing µ-opioid receptors (EC50 = 3 µM). Target: Opioid Receptor. Smiles: COc1ccc(cc1Br)C1SCCN1S(=O)(=O)c1ccc(Cl)cc1. References: Burford NT, et al. Discovery of positive allosteric modulators and silent allosteric modulators of the µ-opioid receptor. Proc Natl Acad Sci U S A. 2013,110(26):10830-10835.
| Keywords: | BMS 986122 |
| Supplier: | TargetMol |
| Supplier-Nr: | T26869 |
Properties
| Application: | µ-opioid receptor positive allosteric modulator |
| MW: | 448.78 D |
| Formula: | C16H15BrClNO3S2 |
Database Information
| CAS : | 313669-88-4| Matching products |
| KEGG ID : | K04215 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
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| H Phrases: | H319 |
| P Phrases: | P264, P280, P305+351+338, P337+313 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
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