Aticaprant

Item number	Size	Delivery time	Price
TGM-TQ0082-1mg	1 mg	7 - 10 business days*	34.00€
TGM-TQ0082-2mg	2 mg	7 - 10 business days*	48.00€
TGM-TQ0082-5mg	5 mg	7 - 10 business days*	81.00€
TGM-TQ0082-1mL	1 ml	7 - 10 business days*	88.00€
TGM-TQ0082-10mg	10 mg	7 - 10 business days*	128.00€
TGM-TQ0082-25mg	25 mg	7 - 10 business days*	271.00€
TGM-TQ0082-50mg	50 mg	7 - 10 business days*	427.00€
TGM-TQ0082-100mg	100 mg	7 - 10 business days*	638.00€

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Description: Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of... more

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Product information "Aticaprant"

Description: Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM). Target: Opioid Receptor. Smiles: Cc1cc(C)cc(c1)[C@@H]1CCCN1Cc1ccc(Oc2ccc(cc2F)C(N)=O)cc1. References: Rorick-Kehn LM, et al. LY2456302 is a novel, potent, orally-bioavailable small molecule kappa-selective antagonist with activity in animal models predictive of efficacy in mood and addictive disorders. Neuropharmacology. 2014 Feb,77:131-44.

Keywords:	LY-2456302, CERC-501
Supplier:	TargetMol
Supplier-Nr:	TQ0082

Properties

Application:	Targets kappa-type opioid receptor (OPRK1)
MW:	418.5 D
Formula:	C26H27FN2O2

Database Information

CAS :	1174130-61-0\| Matching products
KEGG ID :	K04214 \| Matching products

Handling & Safety

Storage:	-20°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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