ARQ 531

Item number	Size	Manual	Delivery time	Price
TGM-T14323-1mg	1 mg	-	7 - 10 business days*	53.00€
TGM-T14323-2mg	2 mg		7 - 10 business days*	74.00€
TGM-T14323-5mg	5 mg		7 - 10 business days*	119.00€
TGM-T14323-1mL	1 ml		7 - 10 business days*	129.00€
TGM-T14323-10mg	10 mg		7 - 10 business days*	201.00€
TGM-T14323-25mg	25 mg		7 - 10 business days*	460.00€
TGM-T14323-50mg	50 mg		7 - 10 business days*	677.00€
TGM-T14323-100mg	100 mg		7 - 10 business days*	966.00€

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Description: ARQ-531 is a potent and orally active BTK inhibitor with potential antineoplastic... more

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Product information "ARQ 531"

Description: ARQ-531 is a potent and orally active BTK inhibitor with potential antineoplastic activity, with IC50s of 0.85 nM and 0.39 nM for WT-BTK and C481S-BTK, respectively. Target: BTK. Smiles: OC[C@@H]1CC[C@H](CO1)Nc1ncnc2[nH]cc(C(=O)c3ccc(Oc4ccccc4)cc3Cl)c12. References: S Eathiraj, et al. Targeting Ibrutinib-Resistant BTK-C481S Mutation with ARQ 531, a Reversible Non-Covalent Inhibitor of BTK. Clinical Lymphoma Myeloma & Leukemia, 2016, 16: S47-S48.

Supplier:	TargetMol
Supplier-Nr:	T14323

Properties

Application:	Targets Bruton agammaglobulinemia tyrosine kinase [EC:2.7.10.2] (BTK)
MW:	478.93 D
Formula:	C25H23ClN4O4

Database Information

CAS :	2095393-15-8\| Matching products
KEGG ID :	K07370 \| Matching products

Handling & Safety

Storage:	+4°C
Shipping:	+4°C (International: +4°C)

Caution
Our products are for laboratory research use only: Not for administration to humans!

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