AM251
If you have any questions, please use our Contact Form.
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
You can also order by e-mail: info@biomol.com
Larger quantity required? Request bulk
Description: AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays... more
Product information "AM251"
Description: AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors, also effective GPR55 agonist (EC50: 39 nM). Target: Cannabinoid Receptor, GPR. Smiles: CC1=C(N(N=C1C(NN2CCCCC2)=O)C3=C(Cl)C=C(Cl)C=C3)C4=CC=C(I)C=C4. References: Liao C, et al. Basic Clin Pharmacol Toxicol, 2004, 94(2), 73-78.
| Supplier: | TargetMol |
| Supplier-Nr: | T1915 |
Properties
| Application: | SR 141716A analog |
| MW: | 555.24 D |
| Formula: | C22H21Cl2IN4O |
Database Information
| CAS : | 183232-66-8| Matching products |
| KEGG ID : | K04277 | Matching products |
Handling & Safety
| Storage: | -20°C |
| Shipping: | +4°C (International: +4°C) |
| Signal Word: | Warning |
| GHS Hazard Pictograms: |
|
| H Phrases: | H315, H319, H335 |
| P Phrases: | P261, P264, P271, P280, P302+352, P304+340, P305+351+338, P312, P321, P332+313, P337+313, P362+364, P403+233, P405, P501 |
Caution
Our products are for laboratory research use only: Not for administration to humans!
Our products are for laboratory research use only: Not for administration to humans!
You will get a certificate here
Viewed