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BMS-986020
Item number: TGM-T4016-100mg
Description: BMS-986020 (AM152) is a selective LPA1 antagonist. Target: LPA Receptor, LPL Receptor. Smiles: C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(cc1)C1(CC1)C(O)=O)c1ccccc1. References: Kihara Y et al. Lysophospholipid receptors in drug discovery. Exp Cell Res. 2015 May 1,333(2):171-7.
| Keywords: | BMS986020, AM152 |
| Application: | LPAR1 antagonist |
| CAS | 1257213-50-5 |
| MW: | 482.53 D |
From 49.00€
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BMS 986020
Item number: Cay22049-1
BMS 986020 is an antagonist of lysophosphatidic acid receptor 1 (LPA1, Kb = 0.0067 µM). It is selective for LPA1 over LPA3 in CHO cells expressing the human receptors (IC50s = 0.3 and >1 µM, respectively). BMS 986020 also inhibits organic anion transporting polypeptide 1B1 (OATP1B1), OATP1B3, the bile salt export...
| Keywords: | 1-[4'-[3-methyl-4-[[[(1R)-1-phenylethoxy]carbonyl]amino]-5-isoxazolyl][1,1'-biphenyl]-4-yl]-cyclopropanecarboxylic acid |
| Application: | LPAR1 antagonist |
| CAS | 1257213-50-5 |
| MW: | 482.5 D |
From 44.00€
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