Zu "K22599" wurden 19 Artikel gefunden!
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Lopinavir
Artikelnummer: TGM-T1623-100mg
Description: Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor effective against HIV protease with the Val 82 mutation. It is less affected by serum protein binding compared to the structurally related drug ritonavir. Target: SARS-CoV, HIV Protease. Smiles:...
| Schlagworte: | ABT-378 |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 192725-17-0 |
| MW: | 628.8 D |
ab 41,00 €
Ritonavir
Artikelnummer: TGM-T1525-100mg
Description: Ritonavir (ABT 538) is a peptidomimetic agent that inhibits both HIV-1 and HIV-2 proteases. Ritonavir is highly inhibited by serum proteins but boosts the effect of other HIV proteases by blocking their degradation by cytochrome P450. Target: SARS-CoV, Apoptosis, HIV Protease. Smiles:...
| Schlagworte: | A 84538, ABT 538, RTV, Abbott 84538 |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 155213-67-5 |
| MW: | 720.94 D |
ab 32,00 €
Brecanavir
Artikelnummer: TGM-T30585-100mg
Description: Brecanavir is a tyrosyl-based arylsulfonamide, high affinity, protease inhibitor (PI) for the treatment of human immunodeficiency virus type 1. Target: Others. Smiles: O(C(N[C@@H](CC1=CC=C(OCC=2N=C(C)SC2)C=C1)[C@@H](CN(S(=O)(=O)C=3C=C4C(=CC3)OCO4)CC(C)C)O)=O)[C@@H]5[C@]6([C@@](OC5)(OCC6)[H])[H]....
| Schlagworte: | CHEMBL206031, UNII-E367I8C7FI, GW-640385X, GW-0385, GW-640385 |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 313682-08-5 |
| MW: | 703.82 D |
ab 1.638,00 €
Palinavir
Artikelnummer: TGM-T28292-100mg
Description: Palinavir is an antiviral, it inhibits HIV-1 protease. Target: Others. Smiles: C([C@H]([C@H](CC1=CC=CC=C1)NC([C@@H](NC(=O)C2=NC3=C(C=C2)C=CC=C3)[C@H](C)C)=O)O)N4[C@H](C(NC(C)(C)C)=O)C[C@H](OCC=5C=CN=CC5)CC4. References: Lamarre D, Croteau G, Wardrop E, Bourgon L, Thibeault D, Clouette C, Vaillancourt M,...
| Schlagworte: | BILA 2011 BS |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 154612-39-2 |
| MW: | 708.89 D |
ab 1.933,00 €
Nelfinavir
Artikelnummer: TGM-T7779-100mg
Description: Nelfinavir (AG1341) is an antiretroviral drug used in the treatment of the human immunodeficiency virus (HIV) (Ki=2 nM). Nelfinavir is a broad-spectrum, anticancer agent. Target: HIV Protease. Smiles: Cc1c(O)cccc1C(=O)N[C@@H](CSc1ccccc1)[C@H](O)CN1C[C@H]2CCCC[C@H]2C[C@H]1C(=O)NC(C)(C)C. References:...
| Schlagworte: | AG1341 |
| Anwendung: | Targets HIV protease [EC:3.4.23.16 3.4.23.47] (PR) |
| CAS | 159989-64-7 |
| MW: | 567.78 D |
ab 36,00 €
COVID-19 Forschung
Ritonavir
Artikelnummer: Cay13872-10
Ritonavir is an HIV protease inhibitor. It inhibits recombinant HIV-1 protease by 79% when used at a concentration of 0.5 nM. It inhibits HIV-13B-induced cell death in MT-4 human T cell leukemia cells (EC50 = 25 nM) as well as cell death induced by HIV-1LAI, HIV-2ROD, and HIV-2EHO in human MT-2 cells (IC50s = 0.045,...
| Schlagworte: | A-84538, ABT-538, NSC 693184, RTV,... |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 155213-67-5 |
| MW: | 720.9 D |
ab 38,00 €
Saquinavir (mesylate)
Artikelnummer: Cay9001893-5
Saquinavir is an HIV protease inhibitor (Kis = 0.12 and 50 = 2 nM). It also inhibits the activity of the severe acute respiratory coronavirus 2 (SARS-CoV-2) main protease (Mpro), also known as 3C-like protease (3CLpro), with an IC50 value of 9.92 µM.Formal Name:...
| Schlagworte: | Ro 31-8959/003,... |
| Anwendung: | HIV protease inhibitor |
| CAS | 149845-06-7 |
| MW: | 767 D |
ab 60,00 €
Tipranavir
Artikelnummer: Cay21028-1
Tipranavir is a potent, orally bioavailable nonpeptidic HIV aspartyl protease inhibitor (Ki = 95%. Formulation: (Request formulation change), A crystalline solid. Solubility: Chloroform: slightly soluble, Methanol: slightly soluble. lambdamax: 254 nm. SMILES:...
| Schlagworte: | PNU-140690,... |
| Anwendung: | HIV protease inhibitor |
| CAS | 174484-41-4 |
| MW: | 602.7 D |
ab 214,00 €
COVID-19 Forschung
Nelfinavir . mesylate
Artikelnummer: AG-CR1-3726-M010
Soluble in DMSO (15mg/ml), DMF (20mg/ml) or ethanol (20mg/ml). Nelfinavir is an orally bioavailable competitive inhibitor of the human immunodeficiency virus. It potently inhibits HIV-1 (Ki=2nM) and HIV-2 protease in vitro. HIV-1 protease is important for the replication of the virus within the cell and the release...
| Schlagworte: | AG-1343, Nelfin, Viracep |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 159989-65-8 |
| MW: | 663.89 D |
ab 55,00 €
COVID-19 Forschung
Saquinavir . mesylate
Artikelnummer: AG-CR1-3727-M010
Soluble in DMSO (10mg/ml). Saquinavir is an antiretroviral inhibitor of the human immunodeficiency virus. It potently inhibits HIV-1 (Ki=0.12nM) and HIV-2 (Ki<0.1nM) protease in vitro. HIV-1 protease is important for the replication of the virus within the cell and the release of mature viral particles from the...
| Schlagworte: | Ro 31-8959 |
| Anwendung: | Antiviral, HIV protease inhibitor |
| CAS | 149845-06-7 |
| MW: | 766.95 D |
ab 55,00 €
Fosamprenavir (calcium salt)
Artikelnummer: Cay21609-1
Fosamprenavir is a prodrug form of the HIV-1 protease inhibitor amprenavir (Cay-15369). It is converted to amprenavir by alkaline phosphatase in the intestinal epithelium. Formulations containing fosamprenavir have been used in the treatment of HIV infections.Formal Name:...
| Schlagworte: | GW 433908G,... |
| Anwendung: | Antiviral, HIV protease inhibitor prodrug |
| CAS | 226700-81-8 |
| MW: | 623.7 D |
ab 34,00 €
Saquinavir-d9
Artikelnummer: Cay28906-1
Saquinavir-d9 is intended for use as an internal standard for the quantification of saquinavir (Cay-9001893) by GC- or LC-MS. Saquinavir is an HIV protease inhibitor (Kis = 0.12 and 50 = 2 nM). It also inhibits the activity of the severe acute respiratory coronavirus 2 (SARS-CoV-2) main protease (Mpro), also known...
| Schlagworte: | (2S)-N1-[(1S,2R)-3-[(3S,4aS,8aS)-3-[[(1,1-di(methyl-d3)ethyl-2,2,2-d3)amino]carbonyl]octahydro-2(1H)-isoquinolinyl]-2-hydr... |
| Anwendung: | GC-MS, LC-MS, Internal standard, Quantification, HIV protease inhibitor |
| CAS | 1356355-11-7 |
| MW: | 679.9 D |
481,00 €