Zu "K15528" wurden 68 Artikel gefunden!
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Fatty Acid Amide Hydrolase (human, recombinant)
Artikelnummer: Cay10010183-100
Fatty acid amide hydrolase (FAAH) is a serine hydrolase with a major role in the hydrolysis of endocannabinoids. It is composed of an N-terminal transmembrane domain, a catalytic domain containing an amidase signature sequence, a polyproline sequence, and a monotopic membrane binding domain. FAAH is localized to...
| Schlagworte: | FAAH, FAAH1, Oleamide hydrolase 1, Oleamide hydrolase 1, Anandamide amidohydrolase 1, Anandamide amidohydrolase 1,... |
| Anwendung: | Enzyme activity |
| MW: | 67,5 kD |
732,00 €
URB597
Artikelnummer: Cay10046-10
URB597 is a potent and selective inhibitor of fatty acid amide hydrolase (FAAH), the enzyme that hydrolyzes anandamide (AEA, Cay-90050) and other simple esters and amides with long unsaturated acyl chains (IC50 = 4.6 nM and 0.5 nM in brain membranes and intact neurons, respectively). URB597 exhibits both...
| Schlagworte: | (3'-(aminocarbonyl)[1,1'-biphenyl]-3-yl)-cyclohexylcarbamate |
| Anwendung: | FAAH inhibitor |
| CAS | 546141-08-6 |
| MW: | 338.4 D |
ab 44,00 €
PHOP
Artikelnummer: Cay71655-100
Fatty acid amide hydrolase (FAAH) is the enzyme responsible for hydrolysis and inactivation of fatty acid amides including anandamide and oleamide. PHOP is a potent FAAH inhibitor, exhibiting Ki values of 0.094 nM and 0.2 nM for the human and rat enzymes, respectively. Using a proteomics approach, PHOP was screened...
| Schlagworte: | CAY10402, Phenyl hexanoyl oxazolopyridine, 1-oxazolo[4,5-b]pyridin-2-yl-6-phenyl-1-hexanone |
| Anwendung: | FAAH inhibitor |
| CAS | 288862-83-9 |
| MW: | 294.4 D |
ab 67,00 €
Anti-Fatty Acid Amide Hydrolase
Artikelnummer: Cay101600-1
Fatty acid amide hydrolase (FAAH) is a serine hydrolase with a major role in the hydrolysis of endocannabinoids. It is composed of an N-terminal transmembrane domain, a catalytic domain containing an amidase signature sequence, a polyproline sequence, and a monotopic membrane binding domain. FAAH is localized to...
| Schlagworte: | Anti-Faah, Anti-Faah1, Anti-Anandamide amidase, Anti-Anandamide amidase, Anti-Oleamide hydrolase 1, Anti-Oleamide... |
| Anwendung: | IHC, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, rat, mouse, ferret |
431,00 €
AM6701
Artikelnummer: TGM-T72020-10mg
Description: AM6701 is a novel highly potent inhibitor of human alpha/beta hydrolase domain 6 (habhd6). Target: Others. Smiles: CN(C)C(=O)n1nnc(Cc2ccc(cc2)-c2ccccc2)n1
| Anwendung: | Anandamide uptake inhibitor |
| CAS | 1010096-65-7 |
| MW: | 307.357 D |
ab 233,00 €
4-Nonylphenylboronic acid
Artikelnummer: TGM-T7688-100mg
Description: 4-Nonylphenylboronic acid is a inhibitor of FAAH. Target: FAAH. Smiles: CCCCCCCCCc1ccc(cc1)B(O)O. References: Minkkila? A , Saario S M , Ka?Sna?Nen H , et al. Discovery of Boronic Acids as Novel and Potent Inhibitors of Fatty Acid Amide Hydrolase[J]. Journal of Medicinal Chemistry, 2008, 51(22):7057-7060.
| Anwendung: | FAAH inhibitor |
| CAS | 256383-45-6 |
| MW: | 248.17 D |
ab 30,00 €
URB937
Artikelnummer: TGM-T8646-100mg
Description: URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM). Target: FAAH. Smiles: NC(=O)c1cccc(c1)-c1cc(OC(=O)NC2CCCCC2)ccc1O. References: Clapper J R , Moreno-Sanz G , Russo R , et al. Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism.[J]. Nature...
| Anwendung: | FAAH inhibitor |
| CAS | 1357160-72-5 |
| MW: | 354.4 D |
ab 42,00 €
(±)17(18)-EpETE-Ethanolamide
Artikelnummer: TGM-T85120-10mg
Description: (±)17(18)-EpETE-Ethanolamide, an omega-3 endocannabinoid epoxide, originates from eicosapentaenoic ethanolamide (EPEA) through cytochrome P450 (CYP) epoxygenases action and is decomposed by soluble epoxide hydrolase (sEH) and fatty acid amide hydrolase (FA, AH). Its endogenous synthesis occurs in...
| Schlagworte: | 17,18-epoxy-Eicosatetraenoic Acid Ethanolamide, (±)17(18)-EpETE-EA, 17,18-EEQ-EA, (±)17,18-EEQ-Ethanolamide |
| Anwendung: | omega-3 endocannabinoid epoxide, soluble epoxide hydrolase (sEH) & FAAH substrate |
| CAS | 2123491-23-4 |
| MW: | 361.52 D |
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FAAH inhibitor 2
Artikelnummer: TGM-T84404-10mg
Description: FAAH Inhibitor 2 (Compound 17b) is an irreversible inhibitor of fatty acid amide hydrolase (FAAH), demonstrating an IC50 value of 0.153 µM [1]. Target: Others. Smiles: C(OC(NCCCCCCC/C=C\CCCCCCCC)=O)C=1C=CC=NC1
| Anwendung: | FAAH inhibitor |
| CAS | 1450603-63-0 |
| MW: | 388.59 D |
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3-Decyl-5,5'-diphenyl-2-thioxo-4-imidazolidinone
Artikelnummer: TGM-T84521-10mg
Description: 3-Decyl-5,5'-diphenyl-2-thioxo-4-imidazolidinone (compound 45), having a pI50 of 5.89, shows promise as an inhibitor of fatty acid amide hydrolase (FAAH). Despite its activity, it demonstrates a lack of affinity for cannabinoid receptors CB(1) and CB(2) [1]. Target: Others. Smiles:...
| Anwendung: | FAAH inhibitor |
| CAS | 875014-22-5 |
| MW: | 408.6 D |
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O-Arachidonoyl glycidol
Artikelnummer: TGM-T84523-10mg
Description: O-Arachidonoyl glycidol (compound 1), a 2-arachidonoylglycerol (2-AG) analog, effectively inhibits the hydrolysis of cytosolic 2-oleoylglycerol (2-OG) with an IC50 value of 4.5 µM, and also blocks 2-OG and anandamide hydrolysis in membrane fractions with IC50 values of 19 µM and 12 µM, respectively [1]....
| Anwendung: | Fatty acid amide hydrolase inhibitor |
| CAS | 439146-24-4 |
| MW: | 360.53 D |
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CAY10435
Artikelnummer: TGM-T84554-10mg
Description: CAY10435, a beta-ketooxazapyridine and selective FAAH inhibitor, exhibits antimicrobial properties. It binds non-competitively to the FAAH of Dictyostelium discoideum, demonstrating a Kd value of 0.57 nM [1] [2]. Target: Others. Smiles: C(CCCCCCCCCCC)(=O)C1=NC=2C(O1)=CC=CN2
| Anwendung: | FAAH inhibitor |
| CAS | 288862-73-7 |
| MW: | 302.41 D |
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