Zu "K05222" wurden 70 Artikel gefunden!
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(Z)-Capsaicin
Artikelnummer: Cay39929-10
(Z)-Capsaicin is an alkaloid that has been found in Capsicum, has diverse biological activities, and is the cis-isomer of capsaicin (Cay-92350, Cay-10010743). It is an agonist of transient receptor potential vanilloid 1 (TRPV1), inducing calcium uptake in CHO cells expressing human TRPV1 (EC50 = 28.2 nM)....
| Schlagworte: | cis-8-methyl-N-Vanillyl-6-nonenamide, cis-Capsaicin, Zucapsaicin, N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methyl-6-nonenamide |
| Anwendung: | Bioactive alkaloid, TRPV1 agonist |
| CAS | 25775-90-0 |
| MW: | 305.4 D |
ab 34,00 €
Capsaicin
Artikelnummer: Cay92350-100
Capsaicin is a terpene alkaloid that has been found in Capsicum and has diverse biological activities. It induces inward currents in HEK293 cells expressing rat transient receptor potential vanilloid 1 (TRPV1, EC50 = 0.64 µM at neutral pH), an effect that can be blocked by the TRPV1 inhibitor A-425619. Capsaicin (10...
| Schlagworte: | N-[(4-hydroxy-3-methoxyphenyl)methyl]-6E-8-methyl-nonenamide |
| CAS | 404-86-4 |
| MW: | 305.4 D |
ab 115,00 €
Mouse TRPV1 (Transient Receptor Potential Cation Channel...
Artikelnummer: ELK-ELK6373.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Mouse TRPV1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Mouse TRPV1. Next,...
| Schlagworte: | TrpV1, Trpv1, OTRPC1, Vanilloid receptor 1, Osm-9-like TRP channel 1, Transient receptor potential cation channel... |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | mouse |
ab 365,00 €
Human TRPV1 (Transient Receptor Potential Cation Channel...
Artikelnummer: ELK-ELK3768.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human TRPV1. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human TRPV1. Next,...
| Schlagworte: | VR1, TrpV1, TRPV1, OTRPC1, Capsaicin receptor, Vanilloid receptor 1, Osm-9-like TRP channel 1, Transient receptor... |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
ab 365,00 €
Capsazepine
Artikelnummer: Cay10007518-1
Transient receptor potential vanilloid type 1 (TRPV1) is a member of the transient receptor potential (TRP) family that is activated or sensitized by a variety of endogenous stimuli as a result of tissue injury and inflammation. TRPV1 is upregulated during inflammation and plays a role in the perception of pain....
| Schlagworte: | N-[2-(4-chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide |
| Anwendung: | TRPV1 antagonist |
| CAS | 138977-28-3 |
| MW: | 376.9 D |
ab 43,00 €
TRPV1-Tat (trifluoroacetate salt)
Artikelnummer: Cay36955-1
TRPV1-Tat is a peptide antagonist of transient receptor potential vanilloid 1 (TRPV1). It consists of amino acids 736-745 from the A-kinase anchor protein (AKAP)-binding domain of TRPV1 and the cell-penetrating peptide sequence from HIV Tat. TRPV1-Tat (200 µM) inhibits currents induced by heat or phorbol...
| Schlagworte: | 736-745-Tat, Transient Receptor Potential Vanilloid 1-Tat,... |
| Anwendung: | Peptide TRPV1 antagonist |
| MW: | 2929.4 D |
ab 35,00 €
SB-452533
Artikelnummer: Cay37379-10
SB-452533 is a transient receptor potential vanilloid 1 (TRPV1) antagonist. It inhibits heat-induced activation of TRPV1 in HEK293 cells expressing the human channel when used at a concentration of 1 µM.Formal Name: N-(2-bromophenyl)-N'-[2-[ethyl(3-methylphenyl)amino]ethyl]-urea. CAS Number: 459429-39-1. Molecular...
| Schlagworte: | N-(2-bromophenyl)-N'-[2-[ethyl(3-methylphenyl)amino]ethyl]-urea |
| Anwendung: | TRPV1 antagonist |
| CAS | 459429-39-1 |
| MW: | 376.3 D |
ab 96,00 €
BCTC
Artikelnummer: Cay10006309-5
The vanilloid receptor 1 (TRPV1) is a ligand-gated ion channel highly expressed on primary nociceptive neurons that respond to a variety of noxious stimuli, including heat, acid, and other chemical irritants. Because disruptions in TRPV1 activity cause reduced thermal nociception and hyperalgesia, this receptor is...
| Schlagworte: | 4-(3-chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide |
| Anwendung: | TRPV1 antagonist |
| CAS | 393514-24-4 |
| MW: | 372.9 D |
ab 56,00 €
Dihydrocapsaicin
Artikelnummer: Cay92355-5
Dihydrocapsaicin is a terpene alkaloid that has been found in Capsicum and has diverse biological activities. It is active against E. faecalis, B. subtilis, S. aureus, P. aeruginosa, K. pneumoniae, E. coli, and C. albicans (MICs = 0.6-10 µg/ml). Dihydrocapsaicin scavenges DPPH (Cay-14805) and ABTS (Cay-27317)...
| Schlagworte: | N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methyl-nonanamide |
| CAS | 19408-84-5 |
| MW: | 307.4 D |
ab 43,00 €
Resiniferatoxin (high purity)
Artikelnummer: AG-CN2-0534-MC05
Isolated from Euphorbia resinifera. Highly potent TRPV1 agonist. Resiniferatoxin (RTX) is a phorbol-related diterpene ester analog of capsaicin. RTX is a highly potent transient receptor potential vanilloid 1 (TRPV1) agonist (Ki=43pM) and acts as a selective modulator of primary afferent neurons. TRPV1 or vanilloid...
| Schlagworte: | RTX, MCP-101 |
| Anwendung: | Highly potent TRPV1 agonist |
| CAS | 57444-62-9 |
| MW: | 628.72 D |
ab 319,00 €
SB-366791
Artikelnummer: Cay11019-5
The transient receptor potential vanilloid type 1 (TRPV1) receptor is a nonselective cation channel gated by noxious heat, protons, and capsaicin. TRPV1 is present in primary sensory neurons and in both central and peripheral sensory nerve terminals and plays a role in thermal and mechanical hyperalgesia. SB-366791...
| Schlagworte: | 3-(4-chlorophenyl)-N-(3-methoxyphenyl)-2-propenamide |
| Anwendung: | TRPV1 antagonist |
| CAS | 472981-92-3 |
| MW: | 287.7 D |
ab 81,00 €
Olvanil
Artikelnummer: Cay90262-50
Olvanil is a structural analog of capsaicin, which is the noxious active component of hot peppers of the Capsicum genus. It is the amide of vanillylamine and oleic acid. Olvanil acts as an agonist at the vanilloid receptor, VR1, inducing desensitization analgesia in rat and mouse models of pain. Olvanil has complex...
| Schlagworte: | N-Vanillyloleamide, NE 19550, N-[(4-hydroxy-3-methoxyphenyl)methyl]-9Z-octadecenamide |
| Anwendung: | Capsaicin analog |
| CAS | 58493-49-5 |
| MW: | 417.6 D |
ab 72,00 €