Zu "K04578" wurden 29 Artikel gefunden!
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Tildacerfont
Artikelnummer: TGM-T26278-10mg
Description: Tildacerfont is an antagonist of CRF1 and reduces the levels of adrenocorticotropic hormone and adrenal androgen. Tildacerfont can be used in studies about congenital adrenal hyperplasia. Target: CRFR. Smiles: CCC(CC)c1cc(C)nc2c(c(C)nn12)-c1sc(nc1Cl)N1CCOCC1. References: Zorrilla EP, Logrip ML, Koob GF....
| Anwendung: | Targets corticotropin releasing hormone receptor 1 (CRHR1) |
| CAS | 1014983-00-6 |
| MW: | 419.97 D |
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Crinecerfont
Artikelnummer: TGM-T31095-100mg
Description: Crinecerfont (SSR-125543) is a selective antagonist of corticotropin-releasing factor 1 receptor (CRF1) and can be used in studies about Classic congenital adrenal hyperplasia. Target: CRFR. Smiles: [C@H](N(CC#C)C1=NC(=C(C)S1)C2=C(Cl)C=C(OC)C(C)=C2)(CC3CC3)C4=CC(F)=C(C)C=C4. References: Philbert J, et...
| Schlagworte: | SSR125543, SSR-125543A, SSR 125543A, SSR125543A, SSR-125543, SSR 125543 |
| Anwendung: | Targets corticotropin releasing hormone receptor 1 (CRHR1) |
| CAS | 752253-39-7 |
| MW: | 483.04 D |
ab 117,00 €
CP 376395
Artikelnummer: TGM-T4329-100mg
Description: CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist. Target: CRFR. Smiles: O(C1=C(C)C=C(C)C=C1C)C2=C(C)C(NC(CC)CC)=CC(C)=N2. References: Chen YL, et al. 2-aryloxy-4-alkylaminopyridines: discovery of novel corticotropin-releasing factor 1...
| Schlagworte: | CP-316311 |
| Anwendung: | Corticotropin-releasing factor receptor 1 (CRFR-1) antagonist |
| CAS | 175140-00-8 |
| MW: | 326.48 D |
ab 37,00 €
Verucerfont
Artikelnummer: TGM-T7361-100mg
Description: Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) . Target: CRFR. Smiles: CC[C@H](Nc1cc(C)nc2c(c(C)nn12)-c1ccc(OC)cc1C)c1nc(C)no1. References: Schwandt M L , Cortes C R , Kwako L E , et al. The CRF1 Antagonist Verucerfont in Anxious Alcohol Dependent Women:...
| Schlagworte: | NBI77860, GSK561679 |
| Anwendung: | Targets corticotropin releasing hormone receptor 1 (CRHR1) |
| CAS | 885220-61-1 |
| MW: | 406.48 D |
ab 58,00 €
Emicerfont
Artikelnummer: TGM-T15214-100mg
Description: Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM). Target: Others. Smiles: COc1ccc(N2CCc3c2nc(C)cc3-n2ccc(n2)N2CCNC2=O)c(C)c1. References: Zorrilla EP, et al. Behavioral, biological, and chemical perspectives on targeting CRF(1) receptor antagonists to treat...
| Schlagworte: | GW876008 |
| Anwendung: | Targets corticotropin releasing hormone receptor 1 (CRHR1) |
| CAS | 786701-13-1 |
| MW: | 404.46 D |
ab 1.971,00 €
Pexacerfont
Artikelnummer: TGM-T16475-1mg
Description: Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor). Target: CRFR. Smiles: CC[C@@H](C)Nc1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C. References: Zhou L, et al. In vitro and in vivo metabolism and pharmacokinetics of...
| Schlagworte: | BMS-562086 |
| Anwendung: | Targets corticotropin releasing hormone receptor 1 (CRHR1) |
| CAS | 459856-18-9 |
| MW: | 340.42 D |
ab 42,00 €
Antalarmin (hydrochloride)
Artikelnummer: Cay15147-5
Corticotropin-releasing hormone (CRH) secreted from the hypothalamus is the major regulator of pituitary corticotropin-release and consequent glucocorticoid secretion. Antalarmin is a selective, nonpeptide antagonist of the CRH receptor 1 (Ki = 1 nM) that, consequently, reduces the release of corticotropin in...
| Schlagworte: | N-butyl-N-ethyl-2,5,6-trimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine, monohydrochloride |
| Anwendung: | CRH receptor 1 antagonist |
| CAS | 220953-69-5 |
| MW: | 415 D |
ab 150,00 €
Anti-CRHR1 / CRF-R (aa 250 - 263), Internal
Artikelnummer: ARG64128.100
Protein function: G-protein coupled receptor for CRH (corticotropin- releasing factor) and UCN (urocortin). Has high affinity for CRH and UCN. Ligand binding causes a conformation change that triggers signaling via guanine nucleotide-binding proteins (G proteins) and down-stream effectors, such as adenylate cyclase....
| Schlagworte: | Anti-CRFR, Anti-CRHR1, Anti-CRFR-1, Anti-CRH-R1, Anti-CRF-R1, Anti-CRF-R-1, Anti-CRH-R-1, Anti-Corticotropin-releasing... |
| Anwendung: | ELISA, ICC, IF, IHC |
| Wirt: | Goat |
| Spezies-Reaktivität: | mouse |
822,00 €
Anti-CRHR1 / CRF-R (aa 107 - 117), Internal
Artikelnummer: ARG64341.100
Protein function: G-protein coupled receptor for CRH (corticotropin- releasing factor) and UCN (urocortin). Has high affinity for CRH and UCN. Ligand binding causes a conformation change that triggers signaling via guanine nucleotide-binding proteins (G proteins) and down-stream effectors, such as adenylate cyclase....
| Schlagworte: | Anti-CRFR, Anti-CRHR1, Anti-CRFR-1, Anti-CRH-R1, Anti-CRF-R1, Anti-CRF-R-1, Anti-CRH-R-1, Anti-Corticotropin-releasing... |
| Anwendung: | ELISA, ICC, IF, WB, IHC (paraffin) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human, mouse |
822,00 €
Human CRHR1 / Corticotropin-releasing factor receptor 2...
Artikelnummer: G-HUFI01072.96
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
641,00 €
Anti-CRF1
Artikelnummer: NSJ-R34530-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Corticotropin releasing hormone receptor 1, CRFR1 Protein function: G-protein coupled receptor for CRH (corticotropin- releasing factor) and UCN (urocortin). Has high affinity for CRH and UCN....
| Schlagworte: | Anti-CRFR, Anti-CRHR1, Anti-CRFR-1, Anti-CRH-R1, Anti-CRF-R1, Anti-CRF-R-1, Anti-CRH-R-1, Anti-Corticotropin-releasing... |
| Anwendung: | IHC, IF, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human, mouse |
790,00 €
Anti-CRF1
Artikelnummer: NSJ-R34787-100UG
0.5 mg/ml in 1X TBS, pH7.3, with 0.5% BSA (US sourced) and 0.02% sodium azide. Additional name(s) for this target protein: Corticotropin releasing hormone receptor 1, CRHR1 Protein function: G-protein coupled receptor for CRH (corticotropin- releasing factor) and UCN (urocortin). Has high affinity for CRH and UCN....
| Schlagworte: | Anti-CRFR, Anti-CRHR1, Anti-CRFR-1, Anti-CRH-R1, Anti-CRF-R1, Anti-CRF-R-1, Anti-CRH-R-1, Anti-Corticotropin-releasing... |
| Anwendung: | WB, ELISA (peptide) |
| Wirt: | Goat |
| Spezies-Reaktivität: | human, mouse |
790,00 €