Zu "K04284" wurden 42 Artikel gefunden!
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YIL781 hydrochloride
Artikelnummer: TGM-T29174-2mg
Description: YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 µM). Target: Others. Smiles: Cl.CC(C)N1CCC[C@H](Cn2c(C)nc3ccc(Oc4ccc(F)cc4)cc3c2=O)C1. References: Moran and Dailey (2009) Gut peptides: targets for antiobesity drug development?...
| Schlagworte: | YIL-781, YIL 781, YIL781, YIL781 HCl |
| Anwendung: | GHS-R1a antagonist |
| CAS | 1640226-17-0 |
| MW: | 445.96 D |
77,00 €
JMV3002
Artikelnummer: TGM-T35793-1mg
Description: JMV3002 is a potent ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro. At 80 µg/kg, JMV3002 inhibits hexarelin-stimulated food intake by up to 98% in rats. It does not induce growth hormone release nor inhibit hexarelin-stimulated growth hormone secretion at a dose of 160 µg/kg in infant...
| Schlagworte: | JMV3002 |
| Anwendung: | Ghrelin receptor antagonist |
| CAS | 925239-03-8 |
| MW: | 586.68 D |
ab 148,00 €
Relamorelin
Artikelnummer: TGM-T34281-100mg
Description: Relamorelin (RM-131), a selective and potent growth hormone-releasing peptide/growth hormone secretagogue receptor (GHSR) agonist, is a potent growth hormone-releasing peptide mimetic with a high affinity for the GHS-1a receptor Relamorelin is a centrally permeable pentapeptide that increases growth...
| Schlagworte: | BIM28131, BIM-28163, RM 131, BIM-28131, BIM 28163, BIM 28131, BIM28163 |
| Anwendung: | Targets growth hormone secretagogue receptor (GHSR) |
| CAS | 661472-41-9 |
| MW: | 790.97 D |
ab 496,00 €
AZ-GHS-22
Artikelnummer: TGM-T37412-10mg
Description: AZ-GHS-22 is an inverse agonist of the growth hormone secretagogue receptor 1a (GHS-R1a), which is also known as the ghrelin receptor.1It binds to GHS-R1a with an IC50value of 0.77 nM. AZ-GHS-22 decreases food intake in mice by 54% in the first two hours after administration of a 100 mg/kg dose. Target:...
| Anwendung: | GHS-R1a inverse agonist |
| CAS | 1143020-91-0 |
| MW: | 621.17 D |
ab 181,00 €
Pralmorelin HCl
Artikelnummer: TGM-T5025L2-25mg
Description: Pralmorelin HCl is regarded as a Growth Hormone Releasing Factor. Target: Others. Smiles: NCCCC[C@@H](C(N)=O)NC([C@@H](CC1=CC=CC=C1)NC([C@@H](NC([C@H](C)NC([C@H](NC([C@H](N)C)=O)CC2=CC3=C(C=CC=C3)C=C2)=O)=O)CC4=CNC5=CC=CC=C45)=O)=O.Cl.Cl. References: Sawada H. [Effect of newly developed analogue of...
| Schlagworte: | Pralmorelin dihydrochloride, WAY-GPA-748 WAY-GPA748, WAY-GPA 748 |
| Anwendung: | Targets growth hormone secretagogue receptor (GHSR) |
| CAS | 158827-34-0 |
| MW: | 890.9 D |
1.520,00 €
AnaMorelin hydrochloride
Artikelnummer: TGM-T7225-100mg
Description: AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay). Target: GHSR. Smiles: Cl.[H][C@](Cc1c[nH]c2ccccc12)(NC(=O)C(C)(C)N)C(=O)N1CCC[C@@](Cc2ccccc2)(C1)C(=O)N(C)N(C)C. References: Pietra C , Takeda Y , Tazawa-Ogata N , et al. Anamorelin...
| Schlagworte: | RC-1291 hydrochloride, ONO-7643 hydrochloride |
| Anwendung: | Targets growth hormone secretagogue receptor (GHSR) |
| CAS | 861998-00-7 |
| MW: | 583.16 D |
ab 31,00 €
Macimorelin acetate
Artikelnummer: TGM-T68276-100mg
Description: Macimorelin Acetate (EP-1572), an orally active growth hormone (GH) secretagogue and a ghrelin receptor (GHSR) agonist, stimulates GH release. It is utilized in research focusing on adult growth hormone deficiency (AGHD) and Cancer Anorexia-Cachexia Syndrome (CACS). Target: Others. Smiles:...
| Schlagworte: | EP-1572 acetate , AEZS-130 acetate, AEZS-130 acetate, EP-1572 acetate , AEZS-130 acetate, EP-1572 acetate |
| Anwendung: | Targets growth hormone secretagogue receptor (GHSR) |
| CAS | 945212-59-9 |
| MW: | 534.61 D |
ab 527,00 €
Ulimorelin
Artikelnummer: TGM-T17202-100mg
Description: Ulimorelin is a ghrelin receptor agonist (EC50: 29 nM and a Ki of 16 nM). Ulimorelin is a prokinetic agent and causes vasorelaxation through competitive antagonist action at alpha1-adrenoceptors. Target: Others. Smiles:...
| Schlagworte: | TZP-101 |
| Anwendung: | Targets growth hormone secretagogue receptor (GHSR) |
| CAS | 842131-33-3 |
| MW: | 538.65 D |
ab 1.671,00 €
PF-5190457
Artikelnummer: TGM-T16508-10mg
Description: PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36). Target: GHSR. Smiles: Cc1cn2cc(CC(=O)N3CCC4(CN(C4)[C@@H]4CCc5cc(ccc45)-c4cc(C)ncn4)CC3)nc2s1. References: Bhattacharya SK, et al. Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor...
| Schlagworte: | PF-05190457 |
| Anwendung: | GHS-R inverse agonist |
| CAS | 1334782-79-4 |
| MW: | 512.67 D |
ab 31,00 €
Anti-GHSR
Artikelnummer: CSB-PA450853.50
Host Species: Rabbit. Isotype: IgG. Buffer: Liquid in PBS containing 50% glycerol, 0.5% BSA and 0.02% sodium azide. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: The antibody was affinity-purified from rabbit antiserum by affinity-chromatography using specific immunogen....
| Schlagworte: | Anti-GHSR, Anti-GHRP, Anti-GHS-R, Anti-Ghrelin receptor, Anti-GH-releasing peptide receptor, Anti-Growth hormone... |
| Anwendung: | ELISA, WB, IHC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
126,00 €
Anti-GHSR
Artikelnummer: CSB-PA545380.100
Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: GHSR. Antigen Species: Human
| Schlagworte: | Anti-GHSR, Anti-GHRP, Anti-GHS-R, Anti-Ghrelin receptor, Anti-GH-releasing peptide receptor, Anti-Growth hormone... |
| Anwendung: | ELISA, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
ab 167,00 €
Anti-GHSR
Artikelnummer: CSB-PA562807.100
Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: GHSR. Antigen Species: Human
| Schlagworte: | Anti-GHSR, Anti-GHRP, Anti-GHS-R, Anti-Ghrelin receptor, Anti-GH-releasing peptide receptor, Anti-Growth hormone... |
| Anwendung: | ELISA, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse, rat |
ab 167,00 €