Zu "K04226" wurden 46 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
Ornipressin Acetate(3397-23-7,free)
Artikelnummer: TGM-TP1049L-100mg
Description: Ornipressin Acetate (POR-8) is a potent vasoconstrictor, hemostatic and renal agent. Target: Others. Smiles: NCCC[C@@H](C(NCC(N)=O)=O)NC([C@@H]1CCCN1C([C@@H]2CSSC[C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N2)=O)CC(N)=O)=O)CCC(N)=O)=O)Cc3ccccc3)=O)Cc4ccc(O)cc4)=O)N)=O)=O.CC(O)=O. References:...
| Schlagworte: | Orpressin, POR-8 |
| Anwendung: | Vasopressin V1A receptor agonist |
| CAS | 914453-98-8 |
| MW: | 1102.25 D |
ab 57,00 €
Conivaptan hydrochloride
Artikelnummer: TGM-T6453-100mg
Description: Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic. Target: Vasopressin Receptor. Smiles: Cl.Cc1nc-2c(CCN(C(=O)c3ccc(NC(=O)c4ccccc4-c4ccccc4)cc3)c3ccccc-23)[nH]1. References: Wada K, et al....
| Schlagworte: | Conivaptan HCl, YM 087, Vaprisol |
| Anwendung: | Targets arginine vasopressin receptor 1A (AVPR1A) |
| CAS | 168626-94-6 |
| MW: | 535.04 D |
ab 38,00 €
Balovaptan
Artikelnummer: TGM-T14494-100mg
Description: Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism. Target: Vasopressin Receptor. Smiles:...
| Schlagworte: | RG7314 |
| Anwendung: | Targets arginine vasopressin receptor 1A (AVPR1A) |
| CAS | 1228088-30-9 |
| MW: | 409.91 D |
ab 60,00 €
RG7713
Artikelnummer: TGM-T4141-100mg
Description: RG7713 (RO 5028442) has been used in trials studying Autistic Disorder. Target: Vasopressin Receptor. Smiles: CN(C)CCn1cc(C(=O)N2CCC3(CC2)OCc2ccccc32)c2ccc(Cl)cc12. References: Ratni H, et al. Discovery of highly selective brain-penetrant vasopressin 1a antagonists for the potential treatment of autism...
| Schlagworte: | RO 5028442 |
| Anwendung: | Brain-penetrant vasopressin V1a receptor antagonist |
| CAS | 920022-47-5 |
| MW: | 437.96 D |
ab 55,00 €
Fuscoside
Artikelnummer: TGM-T4355-100mg
Description: Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist. Target: Vasopressin Receptor. Smiles: CC(=O)NCCCOc1ccc(cc1)C(=O)N1CCC(CC1)N1C(=O)CCc2ccccc12. References: Yamamura Y,etal.PC-21268, an orally effective, nonpeptide vasopressin V1 receptor antagonist.Science. 1991 Apr...
| Schlagworte: | OPC 21268 |
| Anwendung: | Vasopressin V1a/b receptor antagonist |
| CAS | 131631-89-5 |
| MW: | 449.54 D |
ab 52,00 €
Anti-Avpr1a
Artikelnummer: CSB-PA15624A0Rb.100
Host Species: Rabbit. Isotype: IgG. Buffer: Preservative: 0.1mol/L NaCl, 15mmol/L NaN3, PH7.2. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: >95%, Protein G purified. Target Name: Avpr1a. Antigen Species: Rattus norvegicus (Rat)
| Schlagworte: | Anti-V1aR, Anti-Avpr1a, Anti-AVPR V1a, Anti-Vasopressin V1a receptor, Anti-Antidiuretic hormone receptor 1a,... |
| Anwendung: | ELISA, WB, IHC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | rat, mouse |
ab 167,00 €
Anti-AVPR1A
Artikelnummer: CSB-PA572252.100
Host Species: Rabbit. Isotype: IgG. Buffer: Liquid in PBS containing 50% glycerol, 0.5% BSA and 0.02% sodium azide. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: The antibody was affinity-purified from rabbit antiserum by affinity-chromatography using epitope-specific...
| Schlagworte: | Anti-V1aR, Anti-AVPR1, Anti-AVPR1A, Anti-AVPR V1a, Anti-Vasopressin V1a receptor, Anti-Antidiuretic hormone receptor 1a,... |
| Anwendung: | ELISA, WB |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human, mouse |
ab 126,00 €
Vasopressin V1a receptor (Avpr1a), partial, rat, recombinant
Artikelnummer: CSB-RP156244r.1
Organism: Rattus norvegicus (Rat). Source: E.coli. Expression Region: 7-52aa. Protein Length: Partial. Tag Info: N-terminal GST-tagged. Target Protein Sequence: SQDRSVGNSS PWWPLTTEGS NGSQEAARLG EGDSPLGDVR NEELAK. Purity: Greater than 90% as determined by SDS-PAGE. Endotoxin: Not test. Biological Activity: n/a. Form:...
| Schlagworte: | V1aR, Avpr1a, AVPR V1a, Vasopressin V1a receptor, Antidiuretic hormone receptor 1a, Vascular/hepatic-type arginine... |
| Anwendung: | Activity not tested |
| Exprimiert in: | E.coli |
| Ursprungsart: | rat |
| MW: | 31.9 kD |
ab 292,00 €
SR 49059
Artikelnummer: Cay17972-1
SR 49059 is a selective, nonpeptide antagonist of the V1a subtype of the vasopressin receptor (Ki = 1.1-6.3 nM in human). It demonstrates >2 orders of magnitude lower affinity for V1b, V2, and oxytocin receptors and does not exhibit any intrinsic agonist activity. SR 49059 can inhibit arginine vasopressin-induced...
| Schlagworte: | Relcovaptan,... |
| Anwendung: | AVPR1A antagonist |
| CAS | 150375-75-0 |
| MW: | 620.5 D |
ab 67,00 €
Anti-AVPR1A / V1aR
Artikelnummer: NSJ-RQ5565
0.5mg/ml if reconstituted with 0.2ml sterile DI water. Arginine vasopressin receptor 1A(officially called AVPR1A) is one of the three major receptor types forarginine vasopressin(AVPR1BandAVPR2being the others). It belongs to the subfamily of G-protein coupled receptors which includes AVPR1B, V2R and OXT receptors....
| Schlagworte: | Anti-V1aR, Anti-AVPR1, Anti-AVPR1A, Anti-AVPR V1a, Anti-Vasopressin V1a receptor, Anti-Antidiuretic hormone receptor 1a,... |
| Anwendung: | WB, Direct ELISA |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
772,00 €
Argipressin (acetate)
Artikelnummer: Cay24154-1
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle cells and neonatal rat cardiomyocytes, respectively. It also stimulates the intracellular release of...
| Schlagworte: | [Arg8]-Vasopressin, AVP, 8-L-arginine-vasopressin |
| Anwendung: | Vasoconstrictive & antidiuretic peptide hormone |
| CAS | 129979-57-3 |
| MW: | 1084.2 D |
94,00 €
Conivaptan (hydrochloride)
Artikelnummer: Cay23728-10
Conivaptan is an antagonist of the arginine vasopressin (AVP) receptors V1A and V2 (Kis = 0.48 and 3.04 nM for rat liver V1A and kidney V2, respectively). It also competitively inhibits oxytocin binding to rat uterine oxytocin receptors (Ki = 44 nM) but has no effect on AVP binding to anterior pituitary V1B...
| Schlagworte: | YM-087, N-[4-[(4,5-dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1,1'-biphenyl]-2-carboxamide,... |
| Anwendung: | Vasopressin receptor antagonist |
| CAS | 168626-94-6 |
| MW: | 535 D |
ab 94,00 €