Zu "K04213" wurden 56 Artikel gefunden!
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Naltrindole (hydrochloride)
Artikelnummer: Cay9000705-1
Naltrindole is a potent antagonist of the human delta-opioid receptor (Ki = 0.02-0.3 nM), with much lower affinities for kappa- and µ-opioid receptors (Kis = 10-66 and 6-64 nM, respectively). Naltrindole is commonly used to investigate the role of the delta-opioid receptor in signaling responses to test...
| Schlagworte: | (4bS,8R,8aS,14bR)-7-(cyclopropylmethyl)-5,6,7,8,14,14b-hexahydro-4,8-methanobenzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H... |
| Anwendung: | Potent, selective delta-opioid receptor antagonist |
| CAS | 111469-81-9 |
| MW: | 451 D |
ab 45,00 €
BW-180C
Artikelnummer: TGM-TP1905-100mg
Description: BW-180C (DADLE) is a prototypical delta-opioid receptor agonist that also displays activity at the µ-opioid receptor. Displays antinociceptive activity in vivo. Target: Opioid Receptor. Smiles: [C@H](CC1=CC=CC=C1)(C(N[C@H](CC(C)C)C(O)=O)=O)NC(CNC([C@H](NC([C@H](CC2=CC=C(O)C=C2)N)=O)C)=O)=O. References:...
| Schlagworte: | DADLE |
| Anwendung: | Delta-type opioid receptor peptide agonist |
| CAS | 63631-40-3 |
| MW: | 569.65 D |
ab 40,00 €
Levallorphan tartrate
Artikelnummer: TGM-T25690-100mg
Description: Levallorphan tartrate is an opioid antagonist with properties similar to those of NALOXONE. Levallorphan reverses severe opioid-induced respiratory depression but may exacerbate respiratory depression such as that induced by alcohol or other non-opioid central depressants. Target: Others. Smiles:...
| Schlagworte: | Lorfan |
| Anwendung: | Targets mu-type opioid receptor (OPRM1) |
| CAS | 71-82-9 |
| MW: | 433.49 D |
ab 1.520,00 €
Loperamide oxide
Artikelnummer: TGM-T25753-100mg
Description: Loperamide oxide is a prodrug of loperamide, the effective antidiarrheal. Target: Others. Smiles: C(CCN1(=O)CC[C@@](O)(CC1)C2=CC=C(Cl)C=C2)(C(N(C)C)=O)(C3=CC=CC=C3)C4=CC=CC=C4. References: Kamali F, Huang ML. Increased systemic availability of loperamide after oral administration of loperamide and...
| Schlagworte: | R-58425, R58425, R 58425 |
| Anwendung: | Targets mu-type opioid receptor (OPRM1) |
| CAS | 106900-12-3 |
| MW: | 493.04 D |
ab 1.520,00 €
Metkephamid acetate
Artikelnummer: TGM-T25804L-100mg
Description: Metkephamid acetate is a synthetic opioid pentapeptide and derivative of [Met]enkephalin. It shows as a potent agonist of the delta- and µ-opioid receptors with roughly equipotent affinity, and also has similarly high affinity as well as subtype-selectivity for the kappa3-opioid receptor. Target:...
| Schlagworte: | LY 127623, LY127623, LY-127623, Lilly 127623 |
| Anwendung: | Targets delta-type opioid receptor (OPRD1) |
| CAS | 66960-35-8 |
| MW: | 660.79 D |
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ADL-5859
Artikelnummer: TGM-T6175-100mg
Description: ADL-5859 (ADL5859 Hydrochloride) is a selective delta-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor kappa, µ, and little inhibition for the hERG channel. Target: Opioid Receptor. Smiles: Cl.CCN(CC)C(=O)c1ccc(cc1)C1=CC2(CCNCC2)Oc2cccc(O)c12. References: Le Bourdonnec B, et...
| Schlagworte: | ADL5859 Hydrochloride, ADL5859 HCl |
| Anwendung: | delta-opioid receptor agonist |
| CAS | 850173-95-4 |
| MW: | 428.95 D |
ab 45,00 €
ADL5859 (hydrochloride)
Artikelnummer: Cay27796-10
ADL5859 is a delta-opioid receptor agonist (Ki = 0.84 nM). It is selective for delta-opioid receptors over µ-opioid and kappa-opioid receptors exhibiting 32 and 37% inhibition, respectively, in radioligand binding assays when used at a concentration of 10 µM. ADL5859 (3 mg/kg) completely reverses mechanical...
| Schlagworte: | N,N-diethyl-4-(5-hydroxyspiro[2H-1-benzopyran-2,4'-piperidin]-4-yl)-benzamide, monohydrochloride |
| Anwendung: | delta-opioid receptor agonist |
| CAS | 850173-95-4 |
| MW: | 429 D |
ab 158,00 €
Xorphanol mesylate
Artikelnummer: TGM-T35185L-25mg
Description: Xorphanol mesylate is a biochemical. Target: Others. Smiles: S(C)(=O)(=O)O.C[C@@H]1[C@@]2([C@@]3(C=4C(C[C@]2(N(CC5CCC5)CC3)[H])=CC=C(O)C4)CC(=C)C1)[H]. References: Howes JF, Villarreal JE, Harris LS, Essigmann EM, Cowan A. Xorphanol. Drug Alcohol Depend. 1985 Feb,14(3-4):373-80. PubMed PMID: 4039650.
| Schlagworte: | TR5379M, TR-5379M, TR 5379M |
| Anwendung: | Targets delta-type opioid receptor (OPRD1) |
| CAS | 77287-90-2 |
| MW: | 433.6 D |
1.520,00 €
![[Leu5]-Enkephalin](https://www.biomol.com/media/image/13/cf/d4/TGM-T7173-10mg_200x200.png "[Leu5]-Enkephalin")
[Leu5]-Enkephalin
Artikelnummer: TGM-T7173-100mg
Description: [Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of delta-opioid and µ-opioid receptors (Kis = 4.0 and 3.4 nM, respectively). Target: Endogenous Metabolite, Opioid Receptor. Smiles:...
| Schlagworte: | Leu-enkephalin, Leucyl-enkephalin, Leucine enkephalin |
| Anwendung: | Endogenous neuropeptide, delta-opioid receptor agonist, µ-opioid receptor agonist |
| CAS | 58822-25-6 |
| MW: | 555.62 D |
ab 42,00 €
![[Leu5]-Enkephalin TFA(58822-25-6(free bas))](https://www.biomol.com/media/image/d9/20/17/TGM-T7665-1mL_200x200.png "[Leu5]-Enkephalin TFA(58822-25-6(free bas))")
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
Artikelnummer: TGM-T7665-100mg
Description: [Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent delta-receptor ago. Target: Opioid Receptor, Endogenous Metabolite. Smiles: CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O.O=C(O)C(F)(F)F. References: Robert J Cassell , Krishna K...
| Schlagworte: | Leu-enkephalin, Leucyl-enkephalin, Leucine enkephalin |
| Anwendung: | Endogenous neuropeptide, delta-opioid receptor agonist, µ-opioid receptor agonist |
| CAS | 73563-78-7 |
| MW: | 669.64 D |
ab 46,00 €
SNC 80
Artikelnummer: TGM-T8414-10mg
Description: SNC 80 (NIH 10815) is a potent, highly selective and non-peptide delta-opioid receptor agonist, Ki = 1.78 nM, IC50 = 2.73 nM. SNC80 also selectively activates µ-delta heteromer in HEK293 cells with an EC50 of 52.8 nM. SNC80 shows antinociceptive, antihyperalgesic and antidepressant-like effects. SNC80...
| Schlagworte: | NIH 10815, SNC80, Snc-80 |
| Anwendung: | delta-opioid receptor agonist |
| CAS | 156727-74-1 |
| MW: | 449.63 D |
ab 37,00 €
BMS986187
Artikelnummer: TGM-T8991-100mg
Description: BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor. Target: Opioid Receptor. Smiles: Cc1ccccc1COc1ccc(cc1)C1C2=C(CC(C)(C)CC2=O)OC2=C1C(=O)CC(C)(C)C2. References: Livingston K E , Stanczyk M A , Burford N , et al. Pharmacological Evidence for a Putative...
| Anwendung: | Selective positive allosteric delta-opioid Receptor modulator |
| CAS | 684238-37-7 |
| MW: | 470.6 D |
ab 34,00 €