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BIBS 39
BIBS 39

Artikelnummer: TGM-T3178-10mg

Description: BIBS 39 is a novel nonpeptide angiotensin II (AII) receptor antagonist. Target: RAAS. Smiles: CCCCc1nc2ccc(NC(=O)NC3CCCCC3)cc2n1Cc1ccc(cc1)-c1ccccc1C(O)=O. References: Zhang J, et al. Eur J Pharmacol. 1992 Jul 21,218(1):35-41.
Anwendung: AGTR1 / AGTR2 antagonist
CAS 133085-33-3
MW: 524.65 D
ab 37,00 €
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Angiotensin III, human, mouse
Angiotensin III, human, mouse

Artikelnummer: TGM-T7577-100mg

Description: Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA))(3TFA) is an endogenous angiotensin II receptor (AT2R) agonist(IC50s of 0.648 nM). Target: RAAS. Smiles:...
Schlagworte: Angiotensin III, human, mouse(3TFA)
Anwendung: AT1 / AT2 receptor agonist
CAS 13602-53-4
MW: 931.09 D
ab 48,00 €
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AGTR2 Protein, Human, Recombinant (His & SUMO)
AGTR2 Protein, Human, Recombinant (His & SUMO)

Artikelnummer: TGM-TMPH-02268-100ug

Description: Receptor for angiotensin II. Cooperates with MTUS1 to inhibit ERK2 activation and cell proliferation.
Schlagworte: Type-2 angiotensin II receptor, Angiotensin II type-2 receptor, AT2 receptor
MW: 20.8 kD
ab 236,00 €
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PD 123319 ditrifluoroacetate
PD 123319 ditrifluoroacetate

Artikelnummer: TGM-T12381-200mg

Description: PD 123319 (ditrifluoroacetate) is a potent and selective AT2 angiotensin II receptor antagonist with an IC50 of 34 nM. Target: Others. Smiles: OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.CN(C)c1ccc(Cn2cnc3CN([C@@H](Cc23)C(O)=O)C(=O)C(c2ccccc2)c2ccccc2)cc1C. References: Boulay G, et al. Modulation of angiotensin II...
Anwendung: AT2R antagonist
CAS 136676-91-0
MW: 736.66 D
994,00 €
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Buloxibutid
Buloxibutid

Artikelnummer: TGM-T14337-100mg

Description: Buloxibutid (AT2 receptor agonist C21) is a novel and selective small molecule angiotensin II AT2 receptor agonist, exhibiting Ki values of 0.4 nM and 10 µM for AT2 and AT1 receptors, respectively. Target: RAAS. Smiles: CCCCOC(=O)NS(=O)(=O)c1sc(CC(C)C)cc1-c1ccc(Cn2ccnc2)cc1. References: Wan Y, et al....
Schlagworte: AT2 receptor agonist C21
Anwendung: AT2 receptor agonist
CAS 477775-14-7
MW: 475.62 D
ab 42,00 €
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CGP-42112
CGP-42112

Artikelnummer: TGM-T14939-25mg

Description: CGP-42112 is an agonist of the Angiotensin-II subtype 2 receptor (AT2 R). Target: Others. Smiles: CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCCNC(=O)[C@H](CCCNC(N)=N)NC(=O)OCc1ccccc1)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)c1cccnc1)C(O)=O. References: Takekoshi K, et al....
Schlagworte: CGP42112A
Anwendung: Angiotensin II type 2 (AT2) receptor agonist
CAS 127060-75-7
MW: 1052.18 D
1.130,00 €
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Type-2 angiotensin II receptor (AGTR2), partial, human, recombinant
Type-2 angiotensin II receptor (AGTR2), partial, human,...

Artikelnummer: CSB-EP001466HU.1

Organism: Homo sapiens (Human). Source: E.coli. Expression Region: 1-45aa. Protein Length: Partial. Tag Info: N-terminal 6xHis-SUMO-tagged. Target Protein Sequence: MKGNSTLATT SKNITSGLHF GLVNISGNNE STLNCSQKPS DKHLD. Purity: Greater than 90% as determined by SDS-PAGE. Endotoxin: Not test. Biological Activity: n/a....
Schlagworte: AT2, AGTR2, Type-2 angiotensin II receptor, Angiotensin II type-2 receptor, Recombinant Human Type-2 angiotensin II...
Anwendung: Activity not tested
Exprimiert in: E.coli
Ursprungsart: human
MW: 20.8 kD
ab 247,00 €
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Type-2 angiotensin II receptor (Agtr2), partial, rat, recombinant
Type-2 angiotensin II receptor (Agtr2), partial, rat,...

Artikelnummer: CSB-EP001466RA.1

Organism: Rattus norvegicus (Rat). Source: E.coli. Expression Region: 1-45aa. Protein Length: Extracellular Domain. Tag Info: N-terminal GST-tagged. Target Protein Sequence: MKDNFSFAAT SRNITSSLPF DNLNATGTNE SAFNCSHKPA DKHLE. Purity: Greater than 90% as determined by SDS-PAGE. Endotoxin: Not test. Biological...
Schlagworte: AT2, Agtr2, Type-2 angiotensin II receptor, Angiotensin II type-2 receptor, Recombinant Rat Type-2 angiotensin II receptor...
Anwendung: Activity not tested
Exprimiert in: E.coli
Ursprungsart: rat
MW: 31.9 kD
ab 292,00 €
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Type-2 angiotensin II receptor (Agtr2), partial, rat, recombinant
Type-2 angiotensin II receptor (Agtr2), partial, rat,...

Artikelnummer: CSB-YP001466RA.1

Organism: Rattus norvegicus (Rat). Source: Yeast. Expression Region: 1-45aa. Protein Length: Extracellular Domain. Tag Info: N-terminal 6xHis-tagged. Target Protein Sequence: MKDNFSFAAT SRNITSSLPF DNLNATGTNE SAFNCSHKPA DKHLE. Purity: Greater than 90% as determined by SDS-PAGE. Endotoxin: Not test. Biological...
Schlagworte: AT2, Agtr2, Type-2 angiotensin II receptor, Angiotensin II type-2 receptor, Recombinant Rat Type-2 angiotensin II receptor...
Anwendung: Activity not tested
Exprimiert in: Yeast
Ursprungsart: rat
MW: 6.9 kD
ab 347,00 €
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Anti-AGTR2
Anti-AGTR2

Artikelnummer: CSB-PA963716.100

Host Species: Rabbit. Isotype: IgG. Buffer: -20°C, pH7.4 PBS, 0.05% NaN3, 40% Glycerol. Storage: Upon receipt, store at -20°C or -80°C. Avoid repeated freeze. Purification Method: Antigen affinity purification. Target Name: AGTR2. Antigen Species: Human
Schlagworte: Anti-AT2, Anti-AGTR2, Anti-Type-2 angiotensin II receptor, Anti-Angiotensin II type-2 receptor, AGTR 2 antibody, Agtr2...
Anwendung: ELISA, IHC
Wirt: Rabbit
Spezies-Reaktivität: human, mouse, rat
ab 167,00 €
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PD 123319 (trifluoroacetate salt)
PD 123319 (trifluoroacetate salt)

Artikelnummer: Cay16099-5

Angiotensin II is a peptide hormone that regulates blood pressure and fluid balance, contributing to hypertension, atherosclerosis, left ventricular hypertrophy, myocardial infarction, and heart failure. It binds with high affinity to two distinct receptors: AT1R (angiotensin type 1 receptor) and AT2R (angiotensin...
Schlagworte: (6S)-1-[[4-(dimethylamino)-3-methylphenyl]methyl]-5-(2,2-diphenylacetyl)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine-6-ca...
Anwendung: AT2R antagonist
CAS 136676-91-0
MW: 736.7 D
ab 133,00 €
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Anti-AGTR2
Anti-AGTR2

Artikelnummer: 600-401-X82

Anti-AGTR2 Antibody was affinity purified from monospecific antiserum by immunoaffinity chromatography. Cross reactivity with AGTR2 from other sources has not been determined. Protein function: Receptor for angiotensin II. Cooperates with MTUS1 to inhibit ERK2 activation and cell proliferation. [The UniProt Consortium]
Schlagworte: Anti-AT2, Anti-AGTR2, Anti-Type-2 angiotensin II receptor, Anti-Angiotensin II type-2 receptor
Anwendung: ELISA, IHC, WB
Wirt: Rabbit
Spezies-Reaktivität: human, mouse, rat
834,00 €
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