Zu "K04157" wurden 241 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
NEU
Clozapine (hydrochloride)
Artikelnummer: Cay25779-25
Clozapine is a partial agonist of the serotonin (5-HT) receptor subtype 5-HT1A (Ki = 180 nM). It also binds to the 5-HT2A, 5-HT2C, 5-HT3, 5-HT6, and 5-HT7 receptors (Kis = 3.3, 13, 110, 4, and 21 nM, respectively), as well as the histamine H1 and alpha1-adrenergic receptors (Kis = 2.1 and 23 nM, respectively). It...
| Schlagworte: | 8-chloro-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine, dihydrochloride |
| Anwendung: | Atypical antipsychotic, multi-acting receptor targeted antipsychotic (MARTA) |
| CAS | 2711603-38-0 |
| MW: | 399.7 D |
133,00 €
NEU
(+)-Fenfluramine (hydrochloride)
Artikelnummer: Cay39830-100
(+)-Fenfluramine is an agonist of the serotonin (5-HT) receptor subtypes 5-HT2B and 5-HT2C. It induces serotonin release from superfused midbrain synaptosome preparations isolated from wild-type mice, but not 5-HT2B-/- mice, when used at concentrations of 0.5 or 1 µM. (+)-Fenfluramine (3 or 10 mg/kg) reduces food...
| Schlagworte: | Dexfenfluramine, N-ethyl-alpha-methyl-3-(trifluoromethyl)-benzeneethanamine, monohydrochloride |
| Anwendung: | 5-HT2B / 5-HT2C receptor agonist |
| CAS | 3239-45-0 |
| MW: | 267.7 D |
243,00 €
Risperidone (CRM)
Artikelnummer: Cay40163-1
Risperidone (CRM) (Cay-40163) is a certified reference material classified as an atypical antipsychotic. Risperidone has been abused recreationally. Formulations containing risperidone have been used in the treatment of schizophrenia and bipolar disorder. This product is intended for research and forensic...
| Schlagworte: | Apexidone, Psychodal, R 64766,... |
| Anwendung: | Certified reference material, atypical antipsychotic, serotonin-dopamine antagonists (SDA) |
| CAS | 106266-06-2 |
| MW: | 410.5 D |
134,00 €
Paliperidone (CRM)
Artikelnummer: Cay40387-1
Paliperidone (CRM) (Cay-40387) is a certified reference material categorized as an atypical antipsychotic. Paliperidone is an active metabolite of risperidone. It has anticonvulsant, antinociceptive, and antidepressant-like activities in rats. Paliperidone also inhibits apomorphine-induced agitation and stereotypy...
| Schlagworte: | 9-hydroxy Risperidone, RO76477,... |
| Anwendung: | Certified reference material, atypical antipsychotic |
| CAS | 144598-75-4 |
| MW: | 426.5 D |
252,00 €
5-hydroxytryptamine receptor 2C (Htr2c), recombinant...
Artikelnummer: CSB-CF010889MO.100
Organism: Mus musculus (Mouse). Source: in vitro E.coli expression system. Expression Region: 33-459aa. Protein Length: Full Length of Mature Protein. Tag Info: N-terminal 10xHis-tagged. Target Protein Sequence: IVTDTFNSSD GGRLFQFPDG VQNWPALSIV VIIIMTIGGN ILVIMAVSME KKLHNATNYF LMSLAIADML VGLLVMPLSL LAILYDYVWP...
| Schlagworte: | Htr2c, 5ht1c, 5-HT1C, 5-HT2C, 5-HT-2C, 5-HT-1C, 5-HTR2C, Serotonin receptor 2C, 5-hydroxytryptamine receptor 2C,... |
| Anwendung: | Activity not tested |
| Exprimiert in: | E.coli in vitro |
| Ursprungsart: | mouse |
| MW: | 54.6 kD |
ab 1.458,00 €
Clozapine N-oxide
Artikelnummer: LKT-C4759.25
Metabolite of clozapine. It is 5-HT2 serotonin receptor antagonist.
| Anwendung: | 5-HT2 serotonin receptor antagonist |
| CAS | 34233-69-7 |
| MW: | 342,82 D |
ab 274,00 €
Nelotanserin
Artikelnummer: TGM-T7350-100mg
Description: Nelotanserin (APD125) is a potent 5-HT2A inverse agonist(IC50 : 1.7 nM), a moderately potent 5-HT2C partial inverse agonist t(IC50 :79 nM )and a weak 5-HT2B inverse agonistt(IC50 : 791 nM). Target: 5-HT Receptor. Smiles: COc1ccc(NC(=O)Nc2ccc(F)cc2F)cc1-c1c(Br)cnn1C. References: Al-Shamma H A , Anderson...
| Schlagworte: | APD125 |
| Anwendung: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 839713-36-9 |
| MW: | 437.24 D |
ab 34,00 €
lurasidone-d8
Artikelnummer: TGM-TMIH-0313-10mg
Description: lurasidone-d8 is a deuterated compound of lurasidone. Smiles: [2H]C1([2H])N(C[C@@H]2CCCC[C@H]2CN2C(=O)[C@H]3[C@@H]4CC[C@@H](C4)[C@H]3C2=O)C([2H])([2H])C([2H])([2H])N(C2=NSC3=CC=CC=C23)C1([2H])[2H]
| Anwendung: | GC-MS, LC-MS, internal standard |
| CAS | 1132654-54-6 |
| MW: | 500.73 D |
ab 887,00 €
Paliperidone-d4
Artikelnummer: TGM-TMIH-0420-10mg
Description: Paliperidone-d4 is a deuterated compound of Paliperidone. Paliperidone has a CAS number of 144598-75-4. Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older...
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, Dopamine D2/3-receptor / 5-HT2A-receptor antagonist |
| CAS | 1020719-55-4 |
| MW: | 430.51 D |
ab 592,00 €
Quetiapine-d8 Fumarate
Artikelnummer: TGM-TMIJ-0315-1mg
Description: Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression. Smiles:...
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, multiple receptor antagonist |
| CAS | 1185247-12-4 |
| MW: | 507.63 D |
Bitte fragen Sie den aktuellen Preis für diesen Artikel an.
CP-809101
Artikelnummer: TGM-TQ0130-10mg
Description: CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors). Target: 5-HT Receptor. Smiles: O(CC1=CC(Cl)=CC=C1)C=2N=C(C=NC2)N3CCNCC3. References: Higgins GA, Silenieks LB, Lau W, et al. Evaluation of chemically diverse 5-HT2C receptor...
| Anwendung: | Potent 5-HT2C receptor agonist |
| CAS | 479683-64-2 |
| MW: | 304.77 D |
ab 233,00 €
Naftidrofuryl
Artikelnummer: TGM-T25848-100mg
Description: Naftidrofuryl is used in the management of peripheral and cerebral vascular disorders. It is claimed to enhance cellular oxidative capacity and to be spasmolytic. Target: Others. Smiles: C(C(CC1CCCO1)C(OCCN(CC)CC)=O)C=2C3=C(C=CC2)C=CC=C3. References: de Backer TL, Vander Stichele R, Lehert P, Van Bortel...
| Anwendung: | Targets 5-hydroxytryptamine receptor 2 (HTR2) |
| CAS | 31329-57-4 |
| MW: | 383.52 D |
ab 1.671,00 €