Zu "K04150" wurden 56 Artikel gefunden!
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Betazole (hydrochloride)
Artikelnummer: Cay41712-10
Betazole is a histamine H2 receptor agonist. It induces acid secretion in isolated human gastric glands (EC50 = 120 µM), an effect mediated by histamine H2 receptors. Betazole (3-10 mg/kg) increases pepsin and acid levels in gastric juice in dogs.Formal Name: 1H-pyrazole-3-ethanamine, dihydrochloride. CAS Number:...
| Schlagworte: | Ametazole, Gastramine, 1H-pyrazole-3-ethanamine, dihydrochloride |
| Anwendung: | Histamine H2 receptor agonist |
| CAS | 138-92-1 |
| MW: | 184.1 D |
ab 67,00 €
Tiotidine
Artikelnummer: TGM-T13163-1mL
Description: Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium). Target: Others. Smiles: CN\C(NC#N)=N/CCSCc1csc(NC(N)=N)n1. References: Barth H, et al. Structural requirements of imidazole compounds to be inhibitors or activators of histaminemethyltransferase:...
| Schlagworte: | ICI 125211 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 69014-14-8 |
| MW: | 312.42 D |
ab 54,00 €
Niperotidine
Artikelnummer: TGM-T12228-100mg
Description: Niperotidine is an antagonist of histamine H2-receptor. Target: Histamine Receptor. Smiles: CN(C)Cc1ccc(CSCCN\C(NCc2ccc3OCOc3c2)=C\[N+]([O-])=O)o1. References: Gasbarrini G, et al. Acute liver injury related to the use of Niperotidine. J Hepatol. 1997 Sep,27(3):583-6.
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 84845-75-0 |
| MW: | 434.51 D |
ab 1.520,00 €
Famotidine
Artikelnummer: TGM-T1627-2g
Description: Famotidine (MK-208) is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors on the basolateral membrane of parietal cells, famotidine reduces basal and nocturnal gastric acid secretion, thereby decreasing gastric volume,...
| Schlagworte: | MK-208 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 76824-35-6 |
| MW: | 337.45 D |
49,00 €
Nizatidine
Artikelnummer: TGM-T1575-1g
Description: Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity. Target: Histamine Receptor, AChE. Smiles: CN\C(NCCSCc1csc(CN(C)C)n1)=C\[N+]([O-])=O. References: Lin TM, et al. J Pharmacol Exp Ther, 1986, 239(2), 406-410.
| Schlagworte: | Axid, Acinon, Zanizal |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 76963-41-2 |
| MW: | 331.46 D |
30,00 €
Lavoltidine succinate
Artikelnummer: TGM-T32608-25mg
Description: Lavoltidine succinate is a biochemical. Target: Others. Smiles: OC(=O)CCC(O)=O.Cn1nc(CO)nc1NCCCOc1cccc(CN2CCCCC2)c1
| Schlagworte: | AH23844A, AH-23844A, AH 23844A |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 86160-82-9 |
| MW: | 477.562 D |
1.520,00 €
Methantheline Bromide
Artikelnummer: TGM-T33314-100mg
Description: Methantheline Bromide is a synthetic spasmolytic used to relieve cramps or spasms of the stomach, bowel, and bladder. It is also useful for intestinal or gastric ulcers (peptic ulcer disease), intestinal problems, pancreatitis, gastritis, biliary dysmotility, pyloric or urinary problems. Target: Others....
| Schlagworte: | Frenogastrico, Dixamone bromide, Asabaine, Banthine, Methanthelinium bromide |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 53-46-3 |
| MW: | 420.34 D |
ab 1.520,00 €
Dalcotidine
Artikelnummer: TGM-T31195-100mg
Description: Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right...
| Schlagworte: | KU 1257, KU-1257 |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 120958-90-9 |
| MW: | 319.44 D |
ab 142,00 €
Ranitidine
Artikelnummer: TGM-T3610-100mg
Description: Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers. Target: P450, Antibacterial, Histamine Receptor. Smiles: C(N(C)C)C=1OC(CSCCNC(=CN(=O)=O)NC)=CC1. References: Fedorowicz Z. et al,...
| Schlagworte: | HSDB 3925, Ranitidin |
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 66357-35-5 |
| MW: | 314.4 D |
ab 37,00 €
Oxmetidine mesylate
Artikelnummer: TGM-T68587-100mg
Description: Oxmetidine mesylate is an antagonist to Histamine H2 Receptors. Target: Others. Smiles: CS(O)(=O)=O.CS(O)(=O)=O.Cc1nc[nH]c1CSCCNc1ncc(Cc2ccc3OCOc3c2)c(=O)[nH]1
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 84455-52-7 |
| MW: | 591.67 D |
ab 1.520,00 €
Lupitidine hydrochloride
Artikelnummer: TGM-T68799-100mg
Description: Lupitidine hydrochloride inhibits nocturnal acid secretion. Target: Others. Smiles: Cl.Cl.Cl.CN(C)Cc1ccc(CSCCNc2ncc(Cc3ccc(C)nc3)c(=O)[nH]2)o1
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 72716-75-7 |
| MW: | 522.914 D |
ab 1.520,00 €
Impromidine hydrochloride
Artikelnummer: TGM-T68921-100mg
Description: Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies. Target: Histamine Receptor. Smiles: N=C(NCCCC1=CN=CN1)NCCSCC2=C(C)N=CN2.Cl.Cl.Cl. References: Molina E, et al. Use of impromidine to define specific histamine H-2 effects on...
| Anwendung: | Targets histamine receptor H2 (HRH2) |
| CAS | 65573-02-6 |
| MW: | 430.83 D |
ab 257,00 €