- Suchergebnis für K04146
Cookie-Einstellungen
Diese Website benutzt Cookies, die für den technischen Betrieb der Website erforderlich sind und stets gesetzt werden. Andere Cookies, die den Komfort bei Benutzung dieser Website erhöhen, der Direktwerbung dienen oder die Interaktion mit anderen Websites und sozialen Netzwerken vereinfachen sollen, werden nur mit Ihrer Zustimmung gesetzt.
Konfiguration
Technisch erforderlich
Diese Cookies sind für die Grundfunktionen des Shops notwendig.
"Alle Cookies ablehnen" Cookie
"Alle Cookies annehmen" Cookie
Ausgewählter Shop
CSRF-Token
Cookie-Einstellungen
FACT-Finder Tracking
Individuelle Preise
Kundenspezifisches Caching
Session
Währungswechsel
Komfortfunktionen
Diese Cookies werden genutzt um das Einkaufserlebnis noch ansprechender zu gestalten, beispielsweise für die Wiedererkennung des Besuchers.
Facebook-Seite in der rechten Blog - Sidebar anzeigen
Merkzettel
Statistik & Tracking
Endgeräteerkennung
Kauf- und Surfverhalten mit Google Tag Manager
Partnerprogramm
Zu "K04146" wurden 51 Artikel gefunden!
Filter schließen
Filtern nach:
Für die Filterung wurden keine Ergebnisse gefunden!
Artikelnummer: Cay35854-10
U-99194 is a dopamine D3 receptor antagonist (Ki = 160 nM for the human receptor). It is selective for dopamine D3 receptors over the alpha1-adrenergic receptor (alpha1-AR, Ki = 8,913 nM for the rat receptor), M1 muscarinic acetylcholine receptor (mAChR), serotonin (5-HT) receptor subtype 5-HT1A, and dopamine D4...
Schlagworte: | PNU-99194, U-99194A, 2,3-dihydro-5,6-dimethoxy-N,N-dipropyl-1H-inden-2-amine, 2Z-butenedioate |
Anwendung: | Dopamine D3 receptor antagonist |
CAS | 234757-41-6 |
MW: | 393.5 D |
ab 78,00 €
Artikelnummer: ELK-ELK1574.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human DRD3. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human DRD3. Next,...
Schlagworte: | Dopamine D3 receptor, D(3) dopamine receptor |
Anwendung: | ELISA |
Spezies-Reaktivität: | human |
ab 365,00 €
Artikelnummer: Cay16222-50
Pimozide is a dopamine receptor antagonist (Kis = 2.4, 0.3, and 1.8 nM for D2, D3, and D4 receptors, respectively). It also binds to eight additional receptors (Kds = 25-3,100 nM for the human receptors) and inhibits the voltage-gated sodium channel Nav1.2 and the voltage-gated potassium channel Kv11.1 (IC50s = 42...
Schlagworte: | NSC 170984, R 6238, 1-[1-[4,4-bis(4-fluorophenyl)butyl]-4-piperidinyl]-1,3-dihydro-2H-benzimidazol-2-one |
Anwendung: | Dopamine D2/D3-receptor antagonist |
CAS | 2062-78-4 |
MW: | 461.6 D |
ab 43,00 €
Artikelnummer: Cay19530-5
Fluspirilene is a dopamine D2 and D3 receptor antagonist (Kis = 1.5 and 1.1 nM, respectively). It is selective for dopamine D2 and D3 receptors over dopamine D1, alpha1- and alpha2-adrenergic, H1 histamine, and sigma-1 (sigma1) receptors (Kis = 450, 102, >5,000, 540, and 150 nM, respectively), muscarinic...
Schlagworte: | McN-JR 6218, R 6218, Redeptin, 8-[4,4-bis(4-fluorophenyl)butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one |
Anwendung: | Calcium channel blocker, dopamine receptor antagonist |
CAS | 1841-19-6 |
MW: | 475.6 D |
ab 97,00 €
Artikelnummer: Cay14619-25
Amisulpride is a dopamine D2 and D3 receptor antagonist (Kis = 3 and 3.5 nM, respectively). It is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT2B, 5-HT7, and 5-HT7A (Kis = 13, 11.5, and 135.5 nM, respectively). It is selective for these receptors over a panel of 39 additional receptors, ion...
Schlagworte: | DAN 2163, 4-amino-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(ethylsulfonyl)-2-methoxy-benzamide |
Anwendung: | D2 and D3 dopamine receptor antagonist, 5-HT2B and 5-HT7 serotonin receptor antagonist |
CAS | 71675-85-9 |
MW: | 369.5 D |
ab 60,00 €
Artikelnummer: LKT-P6901.25
Is a medication for treating Parkinsons disease and restless leg syndrome. A non-ergoline dopamine agonist.
Schlagworte: | Pramipexole hydrochloride hydrate |
Anwendung: | Dopamine D2/3/4-receptor agonist |
CAS | 104632-25-9 |
MW: | 211,33 D |
ab 135,00 €
Artikelnummer: Cay11982-25
SB 277011A is an antagonist of the dopamine D3 receptor (pKi = 8.0) that is at least 100-fold selective for D3 over other monoamine receptors (pKis = 6.0, 5.0, and 2, 5-HT1D and 5-HT1B respectively). It has high oral bioavailability and enters the central nervous system of the rat. SB 277011A has been shown to have...
Schlagworte: | N-[trans-4-[2-(6-cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide, dihydrochloride |
Anwendung: | DRD3 antagonist |
CAS | 1226917-67-4 |
MW: | 511.5 D |
ab 60,00 €
Artikelnummer: Cay22079-10
PG-01037 is a selective dopamine D3 receptor antagonist (Kis = 0.7, 93, and 375 nM for HEK293 cells expressing human D3, D2, and D4 receptors, respectively). It inhibits quinpirole-induced stimulation of mitogenesis in CHO cells expressing human dopamine D3 receptors (EC50 = 3 nM). PG-01037 (32 mg/kg) reduces...
Schlagworte: | N-[(2E)-4-[4-(2,3-dichlorophenyl)-1-piperazinyl]-2-buten-1-yl]-4-(2-pyridinyl)-benzamide, dihydrochloride |
Anwendung: | DRD3 antagonist |
CAS | 675599-62-9 |
MW: | 554.3 D |
ab 43,00 €
Artikelnummer: Cay21992-25
Dopamine is an endogenous catecholamine neurotransmitter synthesized from the amino acid L-tyrosine that acts as an agonist at dopamine receptors (D1-5). Dopamine is mainly synthesized in the substantia nigra and ventral tegmental area, and is a precursor in norepinephrine and epinephrine biosynthesis....
Schlagworte: | 3-hydroxy Tyramine, DA, KW 3160, 4-(2-aminoethyl)-1,2-benzenediol, monohydrochloride |
Anwendung: | Endogenous catecholamine neurotransmitter |
CAS | 62-31-7 |
MW: | 189.6 D |
123,00 €
Artikelnummer: LKT-S8344.5
Sulpiride is an antipsychotic that functions as an antagonist at D2/3 receptors and also upregulates and activates the GHB receptor. In vivo, sulpiride ameliorates increased impulsivity and attentional impairment in PFC-lesioned models of schizophrenia. Additionally, because dopamine inhibits prolactin release,...
Anwendung: | Dopamine D2-receptor antagonist, Dopamine D3-receptor antagonist |
CAS | 15676-16-1 |
MW: | 341.42 D |
ab 75,00 €
Artikelnummer: NSJ-R30661
0.5mg/ml if reconstituted with 0.2ml sterile DI water. DRD3 is a dopamine receptor that differs in its pharmacology and signaling system from the D1 and D2 receptors and represents both an autoreceptor and a postsynaptic receptor. DRD3 is localized to limbic areas of the brain, which are associated with cognitive,...
Schlagworte: | Anti-DRD3, Anti-Dopamine D3 receptor, Anti-D(3) dopamine receptor, Dopamine Receptor D3 Antibody |
Anwendung: | WB, IHC (paraffin) |
Wirt: | Rabbit |
Spezies-Reaktivität: | human, mouse, rat |
755,00 €
Artikelnummer: Cay21457-1
NGB 2904 is an antagonist that is selective for the dopamine D3 receptor (Ki = 1.4 nM). It potently inhibits quinpirole-stimulated mitogenesis (IC50 = 6.8 nM). NGB 2904 attenuates cocaine- and stress-induced reinstatement of drug-seeking behavior in rats. It also increases spontaneous and amphetamine-stimulated...
Schlagworte: | N-[4-[4-(2,3-dichlorophenyl)-1-piperazinyl]butyl]-9H-fluorene-2-carboxamide, monohydrochloride |
Anwendung: | Dopamine D3 receptor antagonist |
CAS | 189061-11-8 |
MW: | 530.9 D |
ab 53,00 €