Zu "K04145" wurden 144 Artikel gefunden!
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NEU
D (2) dopamine receptor (DRD2), partial, human, recombinant
Artikelnummer: CSB-EP007179HU1.1
Organism: Homo sapiens (Human). Source: E.coli. Expression Region: 214-373aa. Protein Length: Partial. Tag Info: N-terminal 10xHis-tagged and C-terminal Myc-tagged. Target Protein Sequence: IVLRRRRKRV NTKRSSRAFR AHLRAPLKGN CTHPEDMKLC TVIMKSNGSF PVNRRRVEAA RRAQELEMEM LSSTSPPERT RYSPIPPSHH QLTLPDPSHH GLHSTPDSPA...
| Schlagworte: | DRD2, Dopamine D2 receptor, D(2) dopamine receptor, Recombinant Human D (2) dopamine receptor (DRD2), partial |
| Anwendung: | Activity not tested |
| Exprimiert in: | E.coli |
| Ursprungsart: | human |
| MW: | 25.8 kD |
ab 283,00 €
Fluphenazine decanoate
Artikelnummer: Cay39903-10
Fluphenazine decanoate is a prodrug form of the dopamine D1 and D2 receptor antagonist fluphenazine (Cay-23555). It induces random mouth movements in rats, an effect that can be reversed by the dopamine receptor antagonists raclopride (Cay-17422) or SCH 23390 (Cay-15631). Chronic administration of fluphenazine...
| Schlagworte: | NSC 169510, QD-10733, SQ 10,733, decanoic acid,... |
| Anwendung: | Fluphenazine (dopamine D2-receptor antagonist) prodrug form, schizophrenic |
| CAS | 5002-47-1 |
| MW: | 591.8 D |
ab 39,00 €
Metoclopramide
Artikelnummer: Cay39844-10
Metoclopramide is a dual antagonist of the serotonin (5-HT) receptor subtype 5-HT3 and dopamine D2 receptor (IC50s = 308 and 483 nM, respectively). It also reversibly inhibits acetylcholinesterase (AChE) isolated from human postmortem caudate nucleus (Kis = 9.3 and 82 µM for competitive and non-competitive...
| Schlagworte: | 4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-methoxy-benzamide |
| Anwendung: | Dual 5-HT3 / dopamine D2 receptor antagonist |
| CAS | 364-62-5 |
| MW: | 299.8 D |
ab 74,00 €
Human DRD2 (Dopamine Receptor D2) ELISA Kit
Artikelnummer: ELK-ELK2105.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human DRD2. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Human DRD2. Next,...
| Schlagworte: | DRD2, Dopamine D2 receptor, D(2) dopamine receptor |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | human |
ab 365,00 €
Rat DRD2 (Dopamine Receptor D2) ELISA Kit
Artikelnummer: ELK-ELK4579.48
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Rat DRD2. Standards or samples are added to the appropriate microtiter plate wells then with a biotin-conjugated antibody specific to Rat DRD2. Next,...
| Schlagworte: | Drd2, Dopamine D2 receptor, D(2) dopamine receptor |
| Anwendung: | ELISA |
| Spezies-Reaktivität: | rat |
ab 365,00 €
Risperidone
Artikelnummer: Cay13629-10
Risperidone is an atypical antipsychotic that binds to dopamine D2 receptors (Ki = 3 nM) and the serotonin (5-HT) receptor subtype 5-HT2A (Ki = 0.12 nM). It also binds to dopamine D4, alpha1- and alpha2-adrenergic, 5-HT1C, 5-HT1D, and histamine H1 receptors (Kis = 7, 0.81, 7.3, 47, 52, and 2.1 nM, respectively)....
| Schlagworte: | Apexidone, Psychodal, R 64766,... |
| Anwendung: | Receptor antagonist |
| CAS | 106266-06-2 |
| MW: | 410.5 D |
ab 92,00 €
COVID-19 Forschung
Haloperidol
Artikelnummer: Cay12014-100
Haloperidol is a typical antipsychotic and dopamine D2-like receptor antagonist (Kis = 0.6, 0.2, and 22 nM, for D2, D3, and D4 receptors, respectively). It also acts as an inverse agonist at dopamine D2 and D3 receptors (IC50s = 0.8 and 0.6 nM, respectively). Haloperidol also binds to alpha1- and alpha2- adrenergic...
| Schlagworte: | McN-JR 1625, NSC 170973, NSC 615296, R 1625, 4-[4-(4-chlorophenyl)-4-hydroxy-1-piperidinyl]-1-(4-fluorophenyl)-1-butanone |
| Anwendung: | Dopamine D2 receptor antagonist |
| CAS | 52-86-8 |
| MW: | 375.9 D |
ab 43,00 €
Trifluoperazine (hydrochloride)
Artikelnummer: Cay15068-1
Trifluoperazine (TFP) is a phenothiazine compound with anti-adrenergic and anti-dopaminergic actions typical of antipsychotic agents. It antagonizes adrenergic receptors, with selectivity for alpha1 over the alpha2 subtypes (Kis = 24, 653, 163, and 391 nM for alpha1A, alpha2A, alpha2B, and alpha2C, respectively)....
| Schlagworte: | SKF 5019, TFP, 10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoromethyl)-10H-phenothiazine, dihydrochloride |
| Anwendung: | Dopamine receptor D2 antagonist |
| CAS | 440-17-5 |
| MW: | 480.4 D |
ab 43,00 €
Thioridazine (hydrochloride)
Artikelnummer: Cay14400-1
Thioridazine is a typical antipsychotic. It binds to dopamine D2, histamine H1, M3 muscarinic, and alpha1- and alpha2-adrenergic receptors (Kis = 5-341.3 nM), as well as the serotonin (5-HT) receptor subtypes 5-HT1A, 5-HT2A, 5-HT2C, 5-HT6, and 5-HT7 (Kis = 10-180.7 nM). Thioridazine (5 mg/kg) reduces...
| Schlagworte: | Aldazine, NSC 186060, 10-[2-(1-methyl-2-piperidinyl)ethyl]-2-(methylthio)-10H-phenothiazine, monohydrochloride |
| Anwendung: | Dopamine D2-receptor antagonist |
| CAS | 130-61-0 |
| MW: | 407 D |
ab 43,00 €
(-)-Apomorphine (hydrochloride)
Artikelnummer: Cay34222-1
(-)-Apomorphine (hydrochloride) (Cay-34222) is an analytical reference standard categorized as a dopamine receptor agonist. This product is intended for analytical forensic applications. This product is also available as a general research tool (Cay-16094).Formal Name:...
| Schlagworte: | NSC 11442, 5,6,6aR,7-tetrahydro-6-methyl-4H-dibenzo[de,g]quinoline-10,11-diol, monohydrochloride |
| Anwendung: | Analytical reference standard, Dopamine receptor agonist |
| CAS | 314-19-2 |
| MW: | 303.8 D |
ab 134,00 €
Bromocriptine (mesylate)
Artikelnummer: Cay14598-50
Bromocriptine is a dopamine receptor agonist (Kis = 1,659, 12.2, 12.2, 59.7, and 1,691 nM for dopamine D1, D2, D3, D4, and D5 receptors, respectively). It also binds to the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT1D (Kis = 12.9 and 10.7 nM, respectively), as well as alpha1-adrenergic receptors (Kis =...
| Schlagworte: | CB-154, (5alpha)-2-bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)-errgotaman-3',6',18-trione, monomethanesulfonate |
| Anwendung: | Dopamine D2 receptor agonist |
| CAS | 22260-51-1 |
| MW: | 750.7 D |
ab 60,00 €
Aripiprazole
Artikelnummer: LKT-A7034.100
Used for the treatment of schizophrenia. Used for the treatment of acute manic and mixed episodes associated with bipolar disorder, and as an adjunct for the treatment of depression.
| Anwendung: | Metabolic studies |
| CAS | 129722-12-9 |
| MW: | 448,39 D |
ab 130,00 €