Zu "K04137" wurden 52 Artikel gefunden!
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BMY 7378 dihydrochloride
Artikelnummer: TGM-T3046-10mg
Description: BMY 7378 dihydrochloride (BMY7378 HCl) , alpha1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor. Target: Adrenergic Receptor, 5-HT Receptor, Dopamine Receptor. Smiles: Cl.COc1ccccc1N1CCN(CCN2C(=O)CC3(CCCC3)CC2=O)CC1.Cl. References: Cleary L, et al. Auton...
| Schlagworte: | BMY7378 HCl |
| Anwendung: | ADRA2C & ADRA1D antagonist |
| CAS | 21102-95-4 |
| MW: | 458.42 D |
ab 37,00 €
Prazosin-d8
Artikelnummer: TGM-TMIH-0449-1mg
Description: Prazosin-d8 is a deuterated compound of Prazosin. Smiles: [2H]C1([2H])N(C(=O)C2=CC=CO2)C([2H])([2H])C([2H])([2H])N(C2=NC3=C(C=C(OC)C(OC)=C3)C(N)=N2)C1([2H])[2H]
| Anwendung: | GC-MS, LC-MS, internal standard, quantification, antihypertensive agent |
| CAS | 1006717-55-0 |
| MW: | 391.45 D |
ab 228,00 €
ADRA1D Reporter Assay System (human)
Artikelnummer: IB-IB31201
This is an all-inclusive cell-based luciferase reporter assay kit targeting the the Human Adrenoreceptor Alpha 1D (ADRA1D). INDIGO's ADRA1A reporter assay utilizes proprietary mammalian cells that have been engineered to provide constitutive expression of the ADRA1D. In addition to ADRA1D Reporter Cells, this kit...
| Schlagworte: | ADRA1A, ADRA1D, Alpha-1D adrenoceptor, Alpha-1D adrenoreceptor, Alpha-1A adrenergic receptor, Alpha-adrenergic receptor... |
| Anwendung: | Functional activity screening |
| Spezies-Reaktivität: | human |
1.448,00 €
ADRA1D Reporter Assay System (human)
Artikelnummer: IB-IB31202
This is an all-inclusive cell-based luciferase reporter assay kit targeting the the Human Adrenoreceptor Alpha 1D (ADRA1D). INDIGO's ADRA1A reporter assay utilizes proprietary mammalian cells that have been engineered to provide constitutive expression of the ADRA1D. In addition to ADRA1D Reporter Cells, this kit...
| Schlagworte: | ADRA1A, ADRA1D, Alpha-1D adrenoceptor, Alpha-1D adrenoreceptor, Alpha-1A adrenergic receptor, Alpha-adrenergic receptor... |
| Anwendung: | Functional activity screening |
| Spezies-Reaktivität: | human |
3.803,00 €
(-)-Norepinephrine (bitartrate hydrate)
Artikelnummer: Cay16673-250
(-)-Norepinephrine is the endogenous isomer of (±)-norepinephrine (Cay-35580) that acts as a neurotransmitter and hormone and is biosynthesized from dopamine by dopamine beta-hydroxylase. It is an agonist of adrenergic receptors (Ki values are 330, 56, and 740 nM for alpha1, alpha2, and beta1 adrenoceptors,...
| Schlagworte: | Arterenol, Levarterenol, L-Noradrenaline, NE, 4-[(1R)-2-amino-1-hydroxyethyl]-1,2-benzenediol... |
| Anwendung: | Adrenergic receptor agonist, dopamine beta-hydroxylase metabolite |
| CAS | 108341-18-0 |
| MW: | 337.3 D |
ab 44,00 €
Acetylcholine (chloride)
Artikelnummer: Cay23829-5
Acetylcholine is a neurotransmitter that binds to nicotinic and muscarinic acetylcholine receptors (AChRs) in the central and peripheral nervous systems. It mediates motor function at the neuromuscular junction but also has functions in the parasympathetic and sympathetic nervous systems. It is involved in learning...
| Schlagworte: | ACh, 2-(acetyloxy)-N,N,N-trimethyl-ethanaminium, monochloride |
| Anwendung: | alpha1-Adrenergic receptor agonist |
| CAS | 60-31-1 |
| MW: | 181.7 D |
50,00 €
Phentolamine (mesylate)
Artikelnummer: Cay16135-100
Phentolamine is a reversible antagonist of alpha-adrenergic receptors, non-specifically binding all alpha1- and alpha2-adrenoceptors with nanomolar affinities. Formulations containing phentolamine have been used in the treatment of hypertensive emergencies, as well as chronic and emergent pain.Formal Name:...
| Schlagworte: | 3-[[(4,5-dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino]-phenol, monomethanesulfonate |
| Anwendung: | alpha1/2-adrenergic receptor antagonist |
| CAS | 65-28-1 |
| MW: | 377.5 D |
ab 60,00 €
Prazosin (hydrochloride)
Artikelnummer: Cay15023-100
Prazosin is an antagonist of alpha1-adrenergic receptors (alpha1-ARs). It selectively binds to alpha1-ARs with Ki values of 0.2, 0.25, and 0.32 nM for the human recombinant alpha1A-, alpha1B-, and alpha1D-ARs, respectively, over alpha2-ARs (Kis = 340 and 3.7 nM in alpha2A-AR-expressing HT-29 cells and...
| Schlagworte: | CP 12,299-1, NSC 292810, [4-(4-amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-2-furanyl-methanone, monohydrochloride |
| Anwendung: | Antihypertensive agent, melatonin MT3 receptor antagonist |
| CAS | 19237-84-4 |
| MW: | 419.9 D |
ab 43,00 €
Urapidil hydrochloride
Artikelnummer: LKT-U6802.500
White solid. An alpha1-adrenergic antagonist. In addition, it has high affinity and selectivity for central 5-hydroxytryptamine binding sites and inhibits platelet aggregation.
| Anwendung: | alpha1-adrenergic antagonist |
| CAS | 64887-14-5 |
| MW: | 423,93 D |
ab 184,00 €
Synephrine
Artikelnummer: LKT-S9753.1
A biogenic amine present in herbal products and citrus juices. It has antidepressant-like effects by stimulating alpha1-adrenoceptors in mice.
| Anwendung: | alpha-adrenergic receptor agonist |
| CAS | 94-07-5 |
| MW: | 167,21 D |
ab 60,00 €
Methyl 5,6,7,8-Tetradehydro Risperidone
Artikelnummer: Cay17801-10
Risperidone (Cay-13629) is a benzisoxazole derivative used for treating schizophrenia, and also the psychotic, affective, or behavioral symptoms associated with other disorders. Methyl 5,6,7,8-tetradehydro risperidone is used as an internal standard used in the quantitative analysis of risperidone.Formal Name:...
| Schlagworte: | 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-2,7-dimethyl-4H-pyrido[1,2-a]pyrimidin-4-one |
| Anwendung: | Internal standard |
| CAS | 106266-08-4 |
| MW: | 420.5 D |
ab 50,00 €
Risperidone E-oxime
Artikelnummer: Cay22156-10
Risperidone E-oxime is a potential impurity found in commercial preparations of risperidone. Risperidone (Cay-13629) is a longer-acting benzisoxazole derivative used for treating schizophrenia, and also the psychotic, affective, or behavioral symptoms associated with other disorders. This second-generation...
| Schlagworte: | 3-[2-[4-[(E)-(2,4-difluorophenyl)(hydroxyimino)methyl]-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]py... |
| Anwendung: | Potential impurity |
| CAS | 691007-09-7 |
| MW: | 430.5 D |
ab 84,00 €