Zu "K01054" wurden 76 Artikel gefunden!
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Anti-MGLL
Artikelnummer: ATA-HPA011347.100
Polyclonal Antibody against Human MGLL, Gene description: monoglyceride lipase, Alternative Gene Names: HU-K5, MAGL, MGL, Validated applications: ICC, Uniprot ID: Q99685, Storage: Store at +4°C for short term storage. Long time storage is recommended at -20°C. Protein function: Converts monoacylglycerides to free...
| Schlagworte: | Anti-MGL, Anti-MAGL, Anti-HU-K5, Anti-Monoglyceride lipase, Anti-Lysophospholipase-like, Anti-Monoacylglycerol lipase,... |
| Anwendung: | ICC |
| Wirt: | Rabbit |
| Spezies-Reaktivität: | human |
477,00 €
CAY10762
Artikelnummer: TGM-T36498-10mg
Description: CAY10762 is an inhibitor of monoacylglycerol lipase (MAGL, IC50= 34.1 nM) that reduces hydrogen peroxide-induced lactate dehydrogenase (LDH) release from Neuro2a cells at a concentration of 1 µM and increases levels of 2-arachidonoyl glycerol in mouse brain at 10 mg/kg. Target: Others. Smiles:...
| Schlagworte: | CAY10762 |
| Anwendung: | Monoacylglycerol lipase (MGL / MAGL) inhibitor |
| CAS | 2514-37-6 |
| MW: | 255.33 D |
ab 94,00 €
URB754
Artikelnummer: TGM-T37374-100mg
Description: URB754 is a potent and noncompetitive inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 value of 200 nM for the recombinant rat brain enzyme. However, it does not inhibit human recombinant, rat brain, or mouse brain MAGL at concentrations up to 100 µM. There is evidence that the MAGL...
| Anwendung: | Potent noncompetitive monoglyceride lipase (MGL) inhibitor |
| CAS | 86672-58-4 |
| MW: | 266.29 D |
ab 88,00 €
KML29
Artikelnummer: TGM-T4052-100mg
Description: KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor. It has effective inhibition of human/mouse/rat MAGL (IC50: 5.9/15/43 nM). It has not inhibitory for FAAH (IC50 > 50 µM). It also effectively and selectively blocks hydrolysis of 2-arachidonoylglycerol (2-AG) in mice (IC50:...
| Anwendung: | MGLL inhibitor |
| CAS | 1380424-42-9 |
| MW: | 549.42 D |
ab 31,00 €
Pristimerin
Artikelnummer: TGM-T4S1050-100mg
Description: 1. Pristimerin (Celastrol methyl ester) has anticancer activity , treatment with Pristimerin may be a potential strategy for the suppression of hypoxia-induced metastasis through the reversal of hypoxia-induced stem cell characteristics and EMT in cancer cells. 2. Pristimerin down-regulates the...
| Schlagworte: | Celastrol methyl ester |
| Anwendung: | Monoacylglycerol lipase inhibitor |
| CAS | 1258-84-0 |
| MW: | 464.64 D |
ab 34,00 €
MJN110
Artikelnummer: TGM-T5815-100mg
Description: MJN110 (Cravatt Reagent) is a potent and selective MAGL inhibitor. Cravatt Reagent inhibits MAGL (IC50 = 9.1 nM). MJN110(Cravatt Reagent) Produces Opioid-Sparing Effects in a Mouse Neuropathic Pain Model. Target: Lipase. Smiles: Clc1ccc(cc1)C(N1CCN(CC1)C(=O)ON1C(=O)CCC1=O)c1ccc(Cl)cc1. References:...
| Schlagworte: | Cravatt Reagent |
| Anwendung: | MGLL inhibitor |
| CAS | 1438416-21-7 |
| MW: | 462.33 D |
ab 43,00 €
ABX-1431
Artikelnummer: TGM-T5353-100mg
Description: ABX-1431 (Elcubragistat) is a selective and orally available CNS-penetrant monoacylglycerol lipase (MAGL/MGLL) inhibitor (IC50: 14 nM). Target: Lipase. Smiles: FC(F)(F)C(OC(=O)N1CCN(Cc2ccc(cc2N2CCCC2)C(F)(F)F)CC1)C(F)(F)F. References: Cisar JS, et al. Identification of ABX-1431, a Selective Inhibitor of...
| Schlagworte: | Elcubragistat |
| Anwendung: | MAGL inhibitor |
| CAS | 1446817-84-0 |
| MW: | 507.39 D |
ab 31,00 €
JW 618
Artikelnummer: TGM-T84465-10mg
Description: JW 618 is a selective inhibitor of ABHD6, demonstrating inhibition concentrations (IC50 values) of 38 nM for mouse ABHD6 and 13 nM for rat ABHD6, indicating its potent activity across species [1]. Target: Others. Smiles: C(N(C(OC(C(F)(F)F)C(F)(F)F)=O)C)C=1C=C(C=CC1)C=2C=CN=CC2
| Anwendung: | Monoacylglycerol lipase inhibitor |
| CAS | 1416133-88-4 |
| MW: | 392.3 D |
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MGLL Protein, Rat, Recombinant (His)
Artikelnummer: TGM-TMPH-03337-100ug
Description: Converts monoacylglycerides to free fatty acids and glycerol. Hydrolyzes the endocannabinoid 2-arachidonoylglycerol, and thereby contributes to the regulation of endocannabinoid signaling, nociperception and perception of pain. Regulates the levels of fatty acids that serve as signaling molecules and...
| Schlagworte: | Monoglyceride lipase, Monoacylglycerol lipase, Mgll |
| MW: | 34.8 kD |
ab 339,00 €
JZL 184
Artikelnummer: TGM-T6554-100mg
Description: JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 µM for inhibition of MAGL and FAAH in mouse brain membranes respectively. Target: Lipase. Smiles: OC(C1CCN(CC1)C(=O)Oc1ccc(cc1)[N+]([O-])=O)(c1ccc2OCOc2c1)c1ccc2OCOc2c1. References: Long JZ, et al. Nat Chem Biol, 2009, 5(1), 37-44.
| Schlagworte: | JZL184 |
| Anwendung: | Selective, potent monoglyceride lipase (MGL) inhibitor |
| CAS | 1101854-58-3 |
| MW: | 520.49 D |
ab 34,00 €
Monoacylglycerol lipase inhibitor 1
Artikelnummer: TGM-T61294-100mg
Description: Monoacylglycerol lipase inhibitor 1, also known as compound 13 [1], is a potent inhibitor of monoacylglycerol lipase. Target: Others. Smiles: C(N(C)[C@H]1C[C@H](C1)C2=CC=C(C(C)C)C=C2)(=O)[C@@H]3C[C@@]4(C3)NC(=O)OC4
| Anwendung: | Monoacylglycerol lipase (MGLL) inhibitor |
| CAS | 2714570-98-4 |
| MW: | 356.46 D |
ab 1.520,00 €
MAGL-IN-1
Artikelnummer: TGM-T11939-2mg
Description: MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM. Target: Lipase. Smiles: CC(C)c1ccc(cc1)C(=O)C1CCN(CC1)C(=O)c1cc(O)ccc1F. References: Granchi C, et al. Optimization of a Benzoylpiperidine Class Identifies a Highly Potent and Selective Reversible...
| Anwendung: | Monoglyceride lipase (MGLL) inhibitor |
| CAS | 2324160-91-8 |
| MW: | 369.43 D |
34,00 €