Zu "K01049" wurden 222 Artikel gefunden!
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Amplite(TM) Colorimetric Acetylcholinesterase Assay Kit
Artikelnummer: ABD-11400
Acetylcholinesterase, also known as AChE, is an enzyme that degrades (through its hydrolytic activity) the neurotransmitter acetylcholine, producing choline and an acetate group. It is mainly found at neuromuscular junctions and cholinergic synapses in the central nervous system, where its activity serves to...
| Anwendung: | Acetylcholinesterase assays |
279,00 €
NEU
GLN-1062
Artikelnummer: Cay41855-10
GLN-1062 is a neuroprotective agent and prodrug form of galantamine (Cay-17559, Cay-35247), an alkaloid with acetylcholine esterase (AChE) inhibitory and nicotinic acetylcholine (nAChR) potentiating activities. It also is active against M. tuberculosis and M. aurum (MIC = 31.25 µg/ml for both). GLN-1062 decreases...
| Schlagworte: | Benzgalantamine, (4aS,6R,8aS)-6H-benzofuro[3a,3,2-ef][2]benzazepin-6-ol,... |
| Anwendung: | Galantamine (acetylcholinesterase inhibitor) prodrug, neuroprotective agent |
| CAS | 224169-27-1 |
| MW: | 391.5 D |
ab 171,00 €
Curvularin
Artikelnummer: TGM-T13628-5mg
Description: Curvularin ((S)-Curvularin) is a quorum-sensing antagonist of Pseudomonas aeruginosa RhlR extractable from Curvularia lunata, a mycotoxin with anti-inflammatory activity, inhibition of cytokine-induced NO synthase, and inhibition of lipopolysaccharide-induced inflammation in antimyelocytes. study...
| Schlagworte: | (S)-Curvularin |
| Anwendung: | Antibiotic, AChE inhibitor |
| CAS | 10140-70-2 |
| MW: | 292.33 D |
661,00 €
Rivastigmine tartrate
Artikelnummer: TGM-T1628-100mg
Description: Rivastigmine tartrate (SDZ-ENA 713) is a carbamate-derived reversible CHOLINESTE RASEINHIBI TOR that is selective for the CENTRAL NERVOUS SYSTEM and is used for the treatment of DEMENTIA in ALZHEIMER DISEASE and PARKINSON DISEASE. Target: AChR, AChE. Smiles:...
| Schlagworte: | ENA 713, SDZ-ENA 713 |
| Anwendung: | Targets acetylcholinesterase [EC:3.1.1.7] (ACHE) |
| CAS | 129101-54-8 |
| MW: | 400.43 D |
ab 47,00 €
beta-NETA
Artikelnummer: TGM-T14194-1mL
Description: beta-NETA (alpha-NETA) is a stable, noncompetitive, slowly reversible choline acetyltransferase (ChAT) inhibitor with an IC50 of 9 µM and is a potent chemokine-like receptor-1 (CMKLR1) antagonist. beta-NETA has anti-cancer activity[1][2]. beta-NETA weakly inhibits cholinesterase (IC50=84 µM) and...
| Schlagworte: | alpha-NETA |
| Anwendung: | Choline acetyltransferase inhibitor |
| CAS | 31059-54-8 |
| MW: | 369.24 D |
ab 31,00 €
Asoxime dichloride
Artikelnummer: TGM-T14333-10mg
Description: Asoxime dichloride (Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate) is an antagonist to acetylcholine receptors (AChRs) including the nicotinic receptor, alpha7 nAChR. Asoxime dichloride (HI-6) can be used as an antigen and improves vaccination efficacy in the nervous system. Asoxime dichloride...
| Schlagworte: | HI-6, Asoxime (dichloride), Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate |
| Anwendung: | AChE reactivator |
| CAS | 34433-31-3 |
| MW: | 359.21 D |
ab 52,00 €
Dimetacrine
Artikelnummer: TGM-T15132-100mg
Description: Dimetacrine is a useful antidepressant. Target: Others. Smiles: C(CCN(C)C)N1C=2C(C(C)(C)C=3C1=CC=CC3)=CC=CC2. References: Kato H, et al. Comparison of cardiovascular toxicities induced by dimetacrine, imipramine and amitriptyline in isolated guinea pig atria and anesthetized dogs. Jpn J Pharmacol. 1974...
| Schlagworte: | Dimethacrine |
| Anwendung: | Targets acetylcholinesterase [EC:3.1.1.7] (ACHE) |
| CAS | 4757-55-5 |
| MW: | 294.43 D |
ab 1.491,00 €
Itopride free base
Artikelnummer: TGM-T1552L-25mg
Description: Itopride HCl is an AChE inhibitor and dopamine D2 receptor antagonist. It inhibits lower esophageal sphincter relaxation. It also used to treat functional dyspepsia and gastroesophageal reflux disease. Target: Others. Smiles: COC1=CC=C(C=C1OC)C(=O)NCC1=CC=C(OCCN(C)C)C=C1. References: Mohamed HM. A study...
| Schlagworte: | Itopride hydrochloride, HSR-803, HSR803, HSR 803 |
| Anwendung: | Targets dopamine receptor D2 (DRD2) |
| CAS | 122898-67-3 |
| MW: | 358.43 D |
1.491,00 €
Neostigmine methyl sulfate
Artikelnummer: TGM-T1612-100mg
Description: Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase, can not cross the blood-brain barrier, used in the treatment of myasthenia gravis. Target: AChR, AChE. Smiles: c1(cc(ccc1)[N+](C)(C)C)OC(=O)N(C)C.S(=O)(=O)(OC)[O-]. References: Huang TH, et al. Yao Xue Xue Bao....
| Schlagworte: | Hodostin, Syntostigmin, Normastigmin |
| Anwendung: | Targets acetylcholinesterase [EC:3.1.1.7] (ACHE) |
| CAS | 51-60-5 |
| MW: | 334.39 D |
ab 50,00 €
Dimebolin
Artikelnummer: TGM-T21499-1mg
Description: Dimebolin (Latrepirdine) is a 5-HT6 antagonist. Target: 5-HT Receptor. Smiles: CN1CCc2c(C1)c1cc(C)ccc1n2CCc1ccc(C)nc1. References: Schaffhauser H , Mathiasen J R , Dicamillo A , et al. Dimebolin is a 5-HT6 antagonist with acute cognition enhancing activities.[J]. Biochemical Pharmacology, 2009,...
| Schlagworte: | Dimebon, Latrepirdine, Dimebone |
| Anwendung: | Targets acetylcholinesterase [EC:3.1.1.7] (ACHE) |
| CAS | 3613-73-8 |
| MW: | 319.44 D |
ab 58,00 €
Hydroxytacrine maleate
Artikelnummer: TGM-T21556-25mg
Description: Hydroxytacrine maleate (Velnacrine maleate) is a cholinesterase (cholinesterase) inhibitor that enhances memory in rodents and may be used in the study of Alzheimer's dementia of the Alzheimer type (SDAT). Target: AChE. Smiles: C(=C\C(O)=O)\C(O)=O.NC1=C2C(=NC=3C1=CC=CC3)CCCC2O. References: Murphy MF, et...
| Schlagworte: | HP 029 maleate, Velnacrine maleate |
| Anwendung: | Targets acetylcholinesterase [EC:3.1.1.7] (ACHE) |
| CAS | 118909-22-1 |
| MW: | 330.34 D |
ab 31,00 €
Methiocarb
Artikelnummer: TGM-T21464-50mg
Description: Methiocarb, a carbamate pesticide, is used as an insecticide, acaricide, bird repellent, and molluscicide. Methiocarb stimulates cholinergic by inhibiting reversibly acetylcholinesterase activity, making methiocarb a potent neurotoxin. Target: Others. Smiles: O=C(OC=1C=C(C(SC)=C(C1)C)C)NC. References:...
| Schlagworte: | Mercaptodimethur, Mesurol |
| Anwendung: | Carbamate pesticide, AChE inhibitor |
| CAS | 2032-65-7 |
| MW: | 225.31 D |
ab 77,00 €