Zu "920022-47-5" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
RG7713
Artikelnummer: TGM-T4141-100mg
Description: RG7713 (RO 5028442) has been used in trials studying Autistic Disorder. Target: Vasopressin Receptor. Smiles: CN(C)CCn1cc(C(=O)N2CCC3(CC2)OCc2ccccc32)c2ccc(Cl)cc12. References: Ratni H, et al. Discovery of highly selective brain-penetrant vasopressin 1a antagonists for the potential treatment of autism...
| Schlagworte: | RO 5028442 |
| Anwendung: | Brain-penetrant vasopressin V1a receptor antagonist |
| CAS | 920022-47-5 |
| MW: | 437.96 D |
ab 55,00 €
RO5028442
Artikelnummer: Cay31452-10
RO5028442 is a brain-penetrant antagonist of vasopressin V1a receptors (Kis = 1 and 39 nM for the human and mouse receptors, respectively). It is greater than 30,000-fold selective for V1 over V2 receptors, as well as over a panel of 120 receptors, ion channels, and enzymes at 3 µM.Formal Name:...
| Schlagworte: | [6-chloro-1-[2-(dimethylamino)ethyl]-1H-indol-3-yl]spiro[isobenzofuran-1(3H),4'-piperidin]-1'-yl-methanone |
| Anwendung: | Brain-penetrant vasopressin V1a receptor antagonist |
| CAS | 920022-47-5 |
| MW: | 438 D |
ab 78,00 €
