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Elagolix sodium
Artikelnummer: TGM-T5031-100mg
Description: Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively). Target: GNRH Receptor. Smiles: [Na+].COc1cccc(c1F)-c1c(C)n(Cc2c(F)cccc2C(F)(F)F)c(=O)n(C[C@H](NCCCC([O-])=O)c2ccccc2)c1=O. References: Barra F, Scala C, Ferrero S2.Elagolix sodium...
| Schlagworte: | NBI-56418 sodium |
| Anwendung: | Targets gonadotropin-releasing hormone receptor (GNRHR) |
| CAS | 832720-36-2 |
| MW: | 653.57 D |
ab 40,00 €
Elagolix (sodium salt)
Artikelnummer: Cay26534-10
Elagolix is an antagonist of the gonadotropin-releasing hormone receptor (GnRHR, Ki = 0.9 nM in a radioligand binding assay). It is selective for GnRHR over the cytochrome P450 (CYP) isoform CYP3A4 (IC50 = 56 µM) as well as a panel of 100 receptors, ion channels, enzymes, and transporters (IC50s = >10 µM). Elagolix...
| Schlagworte: | 4-[[(1R)-2-[5-(2-fluoro-3-methoxyphenyl)-3-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-3,6-dihydro-4-methyl-2,6-dioxo-1(2... |
| Anwendung: | Gonadotropin-releasing hormone receptor antagonist |
| CAS | 832720-36-2 |
| MW: | 653.6 D |
ab 111,00 €
