Zu "824982-41-4" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
A 784168
Artikelnummer: TGM-T21750-5mg
Description: A-784168, a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1), acts on a ligand-gated nonselective cation channel pivotal in integrating pain stimuli including endogenous lipids, capsaicin, heat, and low pH. It demonstrates commendable central nervous system (CNS) penetration upon...
| Anwendung: | TRPV1 antagonist |
| CAS | 824982-41-4 |
| MW: | 479.4 D |
421,00 €
A-784168
Artikelnummer: Cay32855-1
A-784168 is a transient receptor potential vanilloid 1 (TRPV1) competitive antagonist. It inhibits capsaicin-induced activation of TRPV1 in 1321N1 cells expressing TRPV1 (IC50 = 25 nM for the human receptor). A-784168 is selective for TRPV1 over a panel of 74 neurotransmitter receptors, ion channels, and other TRP...
| Schlagworte: | 3,6-dihydro-3'-(trifluoromethyl)-N-[4-[(trifluoromethyl)sulfonyl]phenyl]-[1(2H),2'-bipyridine]-4-carboxamide |
| Anwendung: | TRPV1 antagonist |
| CAS | 824982-41-4 |
| MW: | 479.4 D |
ab 60,00 €
