Zu "81161-17-3" wurden 2 Artikel gefunden!
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Esmolol hydrochloride
Artikelnummer: TGM-T1503-1mL
Description: Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instances of clinically apparent drug induced liver injury. Target: Mitophagy, Adrenergic Receptor, Autophagy. Smiles:...
| Schlagworte: | ASL8052, Esmolol HCl |
| Anwendung: | Targets adrenergic receptor beta-1 (ADRB1) |
| CAS | 81161-17-3 |
| MW: | 331.15 D |
ab 50,00 €
Esmolol (hydrochloride)
Artikelnummer: Cay22581-10
Esmolol is a beta1-adrenergic receptor (beta1-AR) antagonist. It binds to beta1-ARs (Kd = 100 nM in isolated cardiac myocytes) and is 34-fold selective for beta1- over beta2-ARs. Esmolol also inhibits L-type Ca2+ currents (ICa.L) and the fast Na+ current (INa) in rat cardiac myocytes (IC50s = 50 and 169 µM,...
| Schlagworte: | ASL 8052, 4-[2-hydroxy-3-[(1-methylethyl)amino]propoxy]-benzenepropanoic acid, methyl ester, monohydrochloride |
| Anwendung: | beta1-Adrenergic receptor antagonist |
| CAS | 81161-17-3 |
| MW: | 331.8 D |
ab 43,00 €
