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PF-9366
PF-9366

Artikelnummer: TGM-T5191-10mg

Description: PF-9366 is a human methionine adenosyltransferase 2A (Mat2A) inhibitor with an IC50 of 420 nM and a Kd of 170 nM. Target: Methionine Adenosyltransferase (MAT), Others. Smiles: CN(C)CCc1nnc2cc(-c3ccccc3)c3cc(Cl)ccc3n12. References: Quinlan CL, et al. Targeting S-adenosylmethionine biosynthesis with a...
Anwendung: Methionine adenosyltransferase 2A (Mat2A) inhibitor
CAS 72882-78-1
MW: 350.84 D
ab 54,00 €
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PF-9366
PF-9366

Artikelnummer: Cay30782-25

PF-9366 is an inhibitor of methionine adenosyltransferase 2A (Mat2A, IC50 = 420 nM for S-adenosyl-L-methionine (SAM) production in an enzyme assay). It is selective for Mat2A over a panel of neurotransmitter transporters, phosphodiesterases, ion channels, and G protein-coupled receptors, as well as a panel of 39...
Schlagworte: 7-chloro-N,N-dimethyl-5-phenyl-[1,2,4]triazolo[4,3-a]quinoline-1-ethanamine
Anwendung: Methionine adenosyltransferase 2A (Mat2A) inhibitor
CAS 72882-78-1
MW: 350.8 D
ab 111,00 €
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