Zu "684238-37-7" wurden 2 Artikel gefunden!
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BMS986187
Artikelnummer: TGM-T8991-100mg
Description: BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor. Target: Opioid Receptor. Smiles: Cc1ccccc1COc1ccc(cc1)C1C2=C(CC(C)(C)CC2=O)OC2=C1C(=O)CC(C)(C)C2. References: Livingston K E , Stanczyk M A , Burford N , et al. Pharmacological Evidence for a Putative...
| Anwendung: | Selective positive allosteric delta-opioid Receptor modulator |
| CAS | 684238-37-7 |
| MW: | 470.6 D |
ab 34,00 €
BMS 986187
Artikelnummer: Cay21549-1
BMS 986187 is a positive allosteric modulator of delta-opioid receptors. In the presence of the endogenous delta-opioid receptor agonist leu-enkephalin, BMS 986187 has an average EC50 value of 30 nM for beta-arrestin recruitment, but has little to no activity in the absence of an agonist. It is 100-fold selective...
| Schlagworte: | 3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-9-[4-[(2-methylphenyl)methoxy]phenyl]-1H-xanthene-1,8(2H)-dione |
| Anwendung: | Selective positive allosteric delta-opioid Receptor modulator |
| CAS | 684238-37-7 |
| MW: | 470.6 D |
ab 44,00 €
